SCHEMBL21865069

SCHEMBL21865069

Oc1ccc2c(F)c(N3CCOCC3)ccc2c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.46
HPGD P15428 3/20 0.46
ALDH1A1 P00352 3/20 0.46
ALOX15 P16050 2/20 0.46
GAA P10253 2/20 0.46
CASP1 P29466 1/20 0.46
CASP7 P55210 1/20 0.46
HSD17B10 Q99714 1/20 0.46
PRKDC P78527 2/20 0.44
HSD17B1 P14061 1/20 0.43
HSD17B2 P37059 1/20 0.43
AR P10275 1/20 0.42
NPC1 O15118 2/20 0.41
PIK3CA P42336 3/20 0.40
SMN1; SMN2 Q16637 4/20 0.40
TP53 P04637 1/20 0.40
MAPK1 P28482 1/20 0.40
RAB9A P51151 1/20 0.40
LMNA P02545 3/20 0.40
MAPT P10636 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21865072 0.82 BACE1 (0.43) TSHRHPGDALDH1A1ALOX15GAA
SCHEMBL21865286 0.73 HSD17B1 (0.52) TSHRHPGDALDH1A1CASP1CASP7
SCHEMBL23537930 0.73 SMN1; SMN2 (0.64) TSHRHPGDALDH1A1GAANPC1
SCHEMBL25464794 0.71 ALDH1A1 (0.54) TSHRHPGDALDH1A1ALOX15GAA
SCHEMBL4649483 0.71 MAPT (0.59) TSHRHPGDALDH1A1ALOX15GAA
SCHEMBL21864799 0.71 AOC3 (0.56)
SCHEMBL5616457 0.71 NCF1 (0.52) ALDH1A1HSD17B10PRKDCPIK3CAMAPT
SCHEMBL10706814 0.71 MAPT (0.47) TSHRHPGDALDH1A1ALOX15GAA
SCHEMBL5825846 0.68 LGMN (0.67) TSHRHPGDALDH1A1ALOX15GAA
SCHEMBL6068542 0.68 MAPT (0.53) TSHRHPGDALDH1A1ALOX15GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020063854-A1 QUINOLINE-BASED DERIVATIVES AS VAP-1 INHIBITORS 南京明德新药研发有限公司 2020-04-02 WO disclosed