SCHEMBL2187462

SCHEMBL2187462

N#Cc1ccc(CN2CCN(c3nc(C(=O)N4CCN(c5cccc(C(F)(F)F)c5)CC4)cs3)CC2)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.50
ALDH1A1 P00352 2/20 0.50
KDM4C Q9H3R0 1/20 0.50
TDP1 Q9NUW8 1/20 0.50
LMNA P02545 3/20 0.47
NPSR1 Q6W5P4 3/20 0.47
CYP2D6 P10635 3/20 0.47
HTT P42858 2/20 0.47
USP2 O75604 2/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
MAPT P10636 1/20 0.47
FNTA P49354 1/20 0.46
FNTB P49356 1/20 0.46
TSHR P16473 3/20 0.45
MEN1 O00255 2/20 0.45
KMT2A Q03164 2/20 0.45
MAPK1 P28482 1/20 0.45
HSD17B10 Q99714 1/20 0.45
ATM Q13315 1/20 0.45
POLB P06746 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2187377 0.90 CHRM4 (0.55) KDM4EALDH1A1KDM4CTDP1LMNA
SCHEMBL2187072 0.89 ALDH1A1 (0.52) KDM4EALDH1A1KDM4CTDP1LMNA
SCHEMBL2211193 0.89 KMT2A (0.52) ALDH1A1LMNANPSR1HTTSMN1; SMN2
SCHEMBL2187468 0.88 CHRM4 (0.48) KDM4EALDH1A1KDM4CTDP1LMNA
SCHEMBL2185882 0.85 LMNA (0.60) ALDH1A1LMNANPSR1HTTSMN1; SMN2
SCHEMBL2187381 0.83 STAT3 (0.48) KDM4EALDH1A1KDM4CTDP1LMNA
SCHEMBL2187066 0.82 LMNA (0.58) ALDH1A1LMNANPSR1HTTSMN1; SMN2
SCHEMBL2187566 0.82 CETP (0.48) LMNAUSP2SMN1; SMN2TSHRMEN1
SCHEMBL2188107 0.82 ALDH1A1 (0.57) KDM4EALDH1A1LMNANPSR1HTT
SCHEMBL2188169 0.82 LMNA (0.55) ALDH1A1LMNANPSR1HTTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101031567-B Novel heterocyclic NF-kB inhibitors 4SC Corp.,Ltd. (DE) 2011-12-21 CN disclosed
EP-2343293-A1 NOVEL PIPERIDIN-4-YL-THIAZOLE-CARBOXAMIDE ANALOGUES AS INHIBITORS OF T-CELL PROLIFERATION AND USES THEREOF 4SC AG (DE) 2011-07-13 EP disclosed
CN-101405278-A Novel heterocyclic NF-kB inhibitors 4SC AG (DE) 2009-04-08 CN disclosed
CN-101233119-A Novel heterocyclic nf-kb inhibitors 4SC AG (DE) 2008-07-30 CN disclosed
CN-101031567-A Novel heterocyclic NF-kB inhibitors 4SC AG (DE) 2007-09-05 CN disclosed