SCHEMBL21882367

SCHEMBL21882367

CC(C)(C)OC(=O)NC1CCN(NC(=O)c2ccc(Cl)cn2)CC1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 1/20 0.48
CKS1B P61024 1/20 0.47
SKP1 P63208 1/20 0.47
SKP2 Q13309 1/20 0.47
ATF4 P18848 2/20 0.44
USP30 Q70CQ3 2/20 0.43
CNR1 P21554 1/20 0.43
CNR2 P34972 1/20 0.43
USP14 P54578 1/20 0.42
JAK3 P52333 1/20 0.41
BTK Q06187 1/20 0.41
DRD2 P14416 2/20 0.41
KCNA3 P22001 1/20 0.41
CACNB4 O00305 1/20 0.41
CACNA1A O00555 1/20 0.41
CACNA1G O43497 1/20 0.41
CACNG3 O60359 1/20 0.41
CACNA1F O60840 1/20 0.41
CACNA1H O95180 1/20 0.41
CACNB3 P54284 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29437004 1.00 TRPA1 (0.48) TRPA1CKS1BSKP1SKP2ATF4
SCHEMBL21882080 0.84 ATF4 (0.59) CKS1BSKP1SKP2ATF4CNR1
SCHEMBL29436919 0.84 ATF4 (0.59) CKS1BSKP1SKP2ATF4CNR1
SCHEMBL21819339 0.83 ATF4 (0.47) ATF4CNR1
SCHEMBL23323204 0.81 CKS1B (0.60) CKS1BSKP1SKP2CNR1CNR2
SCHEMBL21819472 0.80 STS (0.52) TRPA1CKS1BSKP1SKP2USP30
SCHEMBL209275 0.79 ATF4 (0.41) TRPA1CKS1BSKP1SKP2ATF4
SCHEMBL21882045 0.77 ATF4 (0.76) ATF4USP14KCNA3SSTR4
SCHEMBL17583173 0.77 GRIN2B (0.52) CKS1BSKP1SKP2CNR1CNR2
SCHEMBL23339865 0.77 CKS1B (0.54) CKS1BSKP1SKP2CNR1CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11166942-B2 Inhibitors of integrated stress response pathway Praxis Biotech LLC (US) 2021-11-09 US disclosed
US-20200101047-A1 INHIBITORS OF INTEGRATED STRESS RESPONSE PATHWAY Praxis Biotech LLC 2020-04-02 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11166942-B2 Inhibitors of integrated stress response pathway ATF4, DDIT3, ATF1 TRPA1 4042/4885CKS1B 388/4885SKP1 2347/4885
US-20200101047-A1 INHIBITORS OF INTEGRATED STRESS RESPONSE PATHWAY ATF4, DDIT3, ATF1 TRPA1 4042/4885CKS1B 388/4885SKP1 2347/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.