SCHEMBL21883415

SCHEMBL21883415

Cc1cc(C#N)nc2ccccc12

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.58
BACE1 P56817 1/20 0.55
KDM4E B2RXH2 7/20 0.50
ALDH1A1 P00352 5/20 0.50
L3MBTL1 Q9Y468 3/20 0.47
LMNA P02545 2/20 0.47
MAPT P10636 3/20 0.47
RAB9A P51151 2/20 0.47
POLB P06746 1/20 0.47
GAA P10253 3/20 0.46
NPFFR1 Q9GZQ6 1/20 0.46
NPFFR2 Q9Y5X5 1/20 0.46
SMN1; SMN2 Q16637 4/20 0.45
HPGD P15428 3/20 0.45
ACHE P22303 1/20 0.45
KMT2A Q03164 2/20 0.44
MEN1 O00255 1/20 0.44
TP53 P04637 1/20 0.44
ADRB1 P08588 1/20 0.43
NCF1 P14598 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3086826 0.81 CYP1A2 (0.58) CYP1A2BACE1KDM4EALDH1A1L3MBTL1
SCHEMBL18024104 0.81 CYP1A2 (0.58) CYP1A2BACE1KDM4EALDH1A1L3MBTL1
SCHEMBL3085385 0.81 CYP1A2 (0.58) CYP1A2BACE1KDM4EALDH1A1L3MBTL1
SCHEMBL3295785 0.79 ALDH1A1 (0.52) KDM4EALDH1A1L3MBTL1LMNAMAPT
SCHEMBL17165889 0.78 KDM4E (0.50) CYP1A2KDM4EALDH1A1L3MBTL1LMNA
SCHEMBL18585567 0.78 KDM4E (0.50) CYP1A2BACE1KDM4EALDH1A1L3MBTL1
SCHEMBL18024098 0.77 CYP1A2 (0.53) CYP1A2BACE1KDM4EALDH1A1L3MBTL1
SCHEMBL28739907 0.77 SMN1; SMN2 (0.57) KDM4EALDH1A1LMNAMAPTPOLB
SCHEMBL28806160 0.76 ACACA (0.50) KDM4EALDH1A1L3MBTL1LMNAMAPT
SCHEMBL18289955 0.76 L3MBTL1 (0.47) CYP1A2KDM4EALDH1A1L3MBTL1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111511731-B Olefin compounds as modulators of the farnesol X receptor 百时美施贵宝公司 2023-05-23 CN claimed
CN-112390755-B Heteroaryl method for amine 中国科学院理化技术研究所 2024-08-02 CN disclosed
CN-113754631-B Heteroaryl method of indole 中国科学院理化技术研究所 2022-08-30 CN disclosed
CN-110256342-B Synthetic method of 2-cyano quinoline derivative 河南省科学院化学研究所有限公司 2022-06-07 CN disclosed
CN-113754631-A Heteroaryl method of indole 中国科学院理化技术研究所 2021-12-07 CN disclosed
CN-112390755-A Method for heteroarylation of amine 中国科学院理化技术研究所 2021-02-23 CN disclosed
WO-2020058290-A1 DRUG CONJUGATE COMPRISING QUINOLINE DERIVATIVES CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (FR) 2020-03-26 WO disclosed
CN-110256342-A A kind of synthetic method of 2- cyano-quinoline derivatives 河南省科学院化学研究所有限公司 2019-09-20 CN disclosed
CN-101139342-A Substituted triazole compound and synthesis method thereof NANJING UNIVERSITY OF TECHNOLOGY (CN) 2008-03-12 CN disclosed