SCHEMBL21884787

SCHEMBL21884787

NC(N)NC(=O)c1nc(-c2ccncc2)ccc1O

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAP2K3 P46734 2/20 0.49
MAPK14 Q16539 1/20 0.48
FTO Q9C0B1 2/20 0.47
EGLN1 Q9GZT9 2/20 0.47
KDM5B Q9UGL1 2/20 0.47
KDM2A Q9Y2K7 2/20 0.47
PRKDC P78527 1/20 0.40
ATR Q13535 1/20 0.40
PARP1 P09874 1/20 0.39
CDC7 O00311 1/20 0.39
KDM6B O15054 1/20 0.38
KDM4C Q9H3R0 1/20 0.38
KDM3A Q9Y4C1 1/20 0.38
MAPT P10636 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
ROCK1 Q13464 9/20 0.37
ROCK2 O75116 7/20 0.37
HDAC1 Q13547 1/20 0.37
HDAC2 Q92769 1/20 0.37
CHUK O15111 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21884393 0.79 MAP2K3 (0.51) MAP2K3MAPK14FTOEGLN1KDM5B
SCHEMBL11907713 0.66 MAP2K3 (0.76) MAP2K3MAPK14PRKDCATRKDM6B
SCHEMBL25376032 0.64 HPGD (0.47) MAP2K3MAPK14FTOEGLN1KDM5B
SCHEMBL29106081 0.63 FTO (0.62) MAP2K3FTOEGLN1KDM5BKDM2A
SCHEMBL21884786 0.62 PDPK1 (0.43) MAPTROCK2CHUK
SCHEMBL10112345 0.62 RAB9A (0.49) MAP2K3MAPK14CDC7MAPTTDP1
SCHEMBL7844018 0.61 FTO (0.58) MAP2K3FTOEGLN1KDM5BKDM2A
SCHEMBL3462574 0.60 ATR (0.68) PRKDCATR
SCHEMBL29106060 0.60 P2RY14 (0.46) FTOEGLN1KDM5BKDM2AMAPT
SCHEMBL14917442 0.60 MAP2K3 (0.61) MAP2K3MAPK14PARP1CDC7MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020061473-A1 SMALL MOLECULES TARGETING MUTANT MAMMALIAN PROTEINS JNANA THERAPEUTICS, INC. (US) 2020-03-26 WO disclosed