SCHEMBL21887490

SCHEMBL21887490

O=C(O)c1ccc(-n2sc(Cl)cc2=O)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KAT2B Q92831 2/20 0.56
CA12 O43570 5/20 0.47
CA9 Q16790 5/20 0.47
CA1 P00915 4/20 0.47
DDAH1 O94760 1/20 0.43
ALDH1A1 P00352 3/20 0.43
KMT2A Q03164 3/20 0.43
KDM4E B2RXH2 2/20 0.43
MAPT P10636 2/20 0.43
TDP1 Q9NUW8 2/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
TSHR P16473 3/20 0.42
ALOX15 P16050 1/20 0.42
DAO P14920 1/20 0.42
CA2 P00918 1/20 0.40
SCN2A Q99250 1/20 0.40
TP53 P04637 1/20 0.40
MEN1 O00255 2/20 0.40
POLB P06746 2/20 0.40
HPGD P15428 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21886954 0.77 KAT2B (0.50) KAT2BCA1CA2
SCHEMBL21814475 0.77 TDP1 (0.52) KAT2BALDH1A1KMT2AMAPTTDP1
SCHEMBL9262493 0.76 MAPT (0.46) CA12CA9CA1ALDH1A1KMT2A
SCHEMBL21886795 0.73 CA12 (0.49) KAT2BCA12CA9CA1DDAH1
SCHEMBL9256085 0.73 PMM2 (0.45) KAT2BCA12CA9CA1ALDH1A1
Terephthalic Acid SCHEMBL31588347 0.66 TSHR (0.92) CA12CA9CA1ALDH1A1SMN1; SMN2
SCHEMBL8506515 0.66 CA12 (0.71) CA12CA9CA1DDAH1KDM4E
Terephthalic Acid SCHEMBL2511919 0.63 TSHR (1.00) CA12CA9CA1ALDH1A1SMN1; SMN2
Terephthalic Acid SCHEMBL175823 0.63 TSHR (1.00) CA12CA9CA1ALDH1A1SMN1; SMN2
Terephthalic Acid SCHEMBL5053781 0.63 TSHR (1.00) CA12CA9CA1ALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020065408-A1 SULFOMALEIMIDE-BASED LINKERS AND CORRESPONDING CONJUGATES PIERRE FABRE MEDICAMENT (FR) 2020-04-02 WO disclosed