SCHEMBL9256085

SCHEMBL9256085

O=C(O)c1ccc(-c2cc(=O)n(-c3ccccc3)s2)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PMM2 O15305 1/20 0.45
IDE P14735 1/20 0.45
MPI P34949 1/20 0.45
PHOSPHO1 Q8TCT1 1/20 0.45
APOBEC3G Q9HC16 1/20 0.45
RXRA P19793 5/20 0.42
RXRB P28702 4/20 0.42
EGFR P00533 1/20 0.41
RXRG P48443 1/20 0.41
BCL2 P10415 1/20 0.41
CA12 O43570 1/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
CA9 Q16790 1/20 0.41
SCN2A Q99250 1/20 0.41
KDM4E B2RXH2 3/20 0.40
ALDH1A1 P00352 3/20 0.40
KMT2A Q03164 3/20 0.40
MAPT P10636 2/20 0.40
TDP1 Q9NUW8 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9262493 0.94 MAPT (0.46) PMM2IDEMPIPHOSPHO1APOBEC3G
SCHEMBL28550660 0.83 KAT2B (0.46) PMM2MPIPHOSPHO1APOBEC3GKDM4E
SCHEMBL21887490 0.73 KAT2B (0.56) RXRARXRBCA12CA1CA2
SCHEMBL9265797 0.73 MYC (0.45) KDM4EALDH1A1KMT2AMAPTTDP1
SCHEMBL28551232 0.70 KAT2B (0.46) PMM2MPIPHOSPHO1APOBEC3GKDM4E
SCHEMBL27816597 0.68 RAB9A (0.63) EGFRKMT2AMEN1POLB
SCHEMBL2346605 0.67 KMO (0.76) RXRARXRBEGFRRXRGBCL2
SCHEMBL29906143 0.67 KMO (0.76) RXRARXRBEGFRRXRGBCL2
Ethane SCHEMBL27330257 0.66 MAPT (0.67) RXRARXRBEGFRRXRGBCL2
SCHEMBL7155730 0.66 EGFR (0.72) EGFRMAPTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5411977-A Substituted 2,5-diaryl-4-isothiazolin-3-ones as antiinflammatory and antithrombotic agents THE DUPONT MERCK PHARMACEUTICAL COMPANY (US) 1995-05-02 US disclosed