SCHEMBL21895486

SCHEMBL21895486

CC(C)C(=O)Nc1ccc2c(=O)[nH]cnc2n1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
XIAP P98170 4/20 0.42
GDA Q9Y2T3 1/20 0.40
BIRC2 Q13490 4/20 0.38
GSK3A P49840 1/20 0.37
GSK3B P49841 1/20 0.37
ADORA2A P29274 2/20 0.36
ADORA3 P0DMS8 1/20 0.36
ADORA1 P30542 1/20 0.36
SRC P12931 1/20 0.36
ALDH1A1 P00352 5/20 0.36
RAB9A P51151 4/20 0.36
NPC1 O15118 3/20 0.36
TP53 P04637 2/20 0.36
CHEK1 O14757 1/20 0.36
PARP1 P09874 1/20 0.36
PIM1 P11309 1/20 0.36
RPS6KA3 P51812 1/20 0.36
SLC2A1 P11166 1/20 0.36
KDM4E B2RXH2 2/20 0.36
LMNA P02545 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19699476 0.82 XIAP (0.39) XIAPBIRC2ADORA2AADORA3ADORA1
SCHEMBL29329931 0.73 SMN1; SMN2 (0.40) GSK3AGSK3BADORA2ASRCALDH1A1
SCHEMBL18237704 0.72 PARP1 (0.42) GSK3AGSK3BADORA2ASRCALDH1A1
SCHEMBL1965199 0.70 ADORA3 (0.43) XIAPBIRC2ADORA2AADORA3ADORA1
SCHEMBL19153800 0.70 PARP1 (0.50) ADORA2AADORA1SRCALDH1A1RAB9A
SCHEMBL735411 0.69 GDA (0.72) GDAXDH
SCHEMBL30979186 0.66 PARP1 (0.46) GSK3AGSK3BADORA2ASRCALDH1A1
SCHEMBL21808624 0.66 PARP1 (0.46) GSK3AGSK3BADORA2ASRCALDH1A1
SCHEMBL21339749 0.66 SRC (0.52) ADORA2AADORA1SRCALDH1A1RAB9A
SCHEMBL17776531 0.65 GDA (0.46) GDAADORA3ADORA1KDM4ELMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3854799-B1 CYCLIC DINUCLEOTIDE ANALOGUE, PHARMACEUTICAL COMPOSITION THEREOF, AND APPLICATION SHANGHAI DE NOVO PHARMATECH CO LTD (CN) 2024-07-17 EP disclosed
EP-3854799-A1 CYCLIC DINUCLEOTIDE ANALOGUE, PHARMACEUTICAL COMPOSITION THEREOF, AND APPLICATION Shanghai de Novo Pharmatech Co., Ltd. (CN) 2021-07-28 EP disclosed
WO-2020057546-A1 CYCLIC DINUCLEOTIDE ANALOGUE, PHARMACEUTICAL COMPOSITION THEREOF, AND APPLICATION 上海迪诺医药科技有限公司 2020-03-26 WO disclosed