SCHEMBL1965199

SCHEMBL1965199

CC(C)C(=O)Nc1cc[nH]c(=O)n1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 2/20 0.43
ADORA1 P30542 2/20 0.43
ADORA2A P29274 1/20 0.43
BIRC2 Q13490 4/20 0.41
XIAP P98170 3/20 0.41
ALDH1A1 P00352 7/20 0.40
GAA P10253 1/20 0.40
KDM4E B2RXH2 3/20 0.40
GLA P06280 1/20 0.40
TP53 P04637 2/20 0.39
MDM4 O15151 1/20 0.39
MEN1 O00255 3/20 0.38
KMT2A Q03164 3/20 0.38
HPGD P15428 2/20 0.38
SCN10A Q9Y5Y9 1/20 0.38
MAPT P10636 1/20 0.38
RXFP1 Q9HBX9 1/20 0.38
LMNA P02545 2/20 0.37
HSD17B10 Q99714 1/20 0.37
NPC1 O15118 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3460188 0.83 XIAP (0.36) BIRC2XIAPALDH1A1GAARAB9A
SCHEMBL5667925 0.82 BIRC2 (0.35) ADORA3ADORA1ADORA2ABIRC2XIAP
SCHEMBL21187 0.80 KDM4E (0.47) ADORA3ADORA1ADORA2AKDM4EMAPT
Methane SCHEMBL27916786 0.79 KDM4E (0.46) ADORA3ADORA1ADORA2AKDM4EMAPT
SCHEMBL1827089 0.79 KDM4E (0.46) ADORA3ADORA1ADORA2AKDM4EMAPT
SCHEMBL10679044 0.78 GRM5 (0.36) ADORA1ADORA2AKDM4EMEN1KMT2A
SCHEMBL27342109 0.78 MAOB (0.53) ADORA3ADORA1ADORA2ABIRC2XIAP
SCHEMBL3187090 0.78 SMN1; SMN2 (0.52) ALDH1A1GAAKDM4EMEN1KMT2A
SCHEMBL513900 0.77 CYP3A4 (0.38) ALDH1A1GAAKDM4EMEN1KMT2A
SCHEMBL8709449 0.76 L3MBTL1 (0.46) ADORA1ALDH1A1KDM4ETP53MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 45 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2026106497-A2 FUNCTIONALIZED CIRCULAR RNA AND METHODS AND INTERMEDIATES FOR THEIR PRODUCTION SIEĆ BADAWCZA ŁUKASIEWICZ – PORT POLSKI OSRODEK ROZWOJU TECHNOLOGII (PL) 2026-05-21 WO claimed
US-11180756-B2 Morpholino modified oligomeric compounds Ionis Pharmaceuticals (US) 2021-11-23 US claimed
US-20200239881-A1 MORPHOLINO MODIFIED OLIGOMERIC COMPOUNDS IONIS PHARMACEUTICALS, INC. (US) 2020-07-30 US claimed
US-10287313-B2 RNA monomers containing 0-acetal levulinyl ester groups and their use in RNA microarrays THE ROYAL INSTITUTION FOR THE ADVANCEMENT OF LEARNING/MCGILL UNIVERSITY (CA) 2019-05-14 US claimed
WO-2018165564-A1 MORPHOLINO MODIFIED OLIGOMERIC COMPOUNDS IONIS PHARMACEUTICALS, INC. (US) 2018-09-13 WO claimed
US-20160340382-A1 RNA MONOMERS CONTAINING O-ACETAL LEVULINYL ESTER GROUPS AND THEIR USE IN RNA MICROARRAYS THE ROYAL INSTITUTION FOR THE ADVANCEMENT OF LEARNING/MCGILL UNIVERSITY (CA) 2016-11-24 US claimed
EP-2334692-B1 RNA MONOMERS CONTAINING O-ACETAL LEVULINYL ESTER GROUPS AND THEIR USE IN RNA MICROARRAYS UNIV MCGILL (CA) 2016-04-13 EP claimed
US-9249175-B2 RNA monomers containing O-acetal levulinyl ester groups and their use in RNA microarrays THE ROYAL INSTITUTE FOR THE ADVANCEMENT OF LEARNING/MCGILL UNIVERSITY (CA) 2016-02-02 US claimed
US-20120178638-A1 RNA MONOMERS CONTAINING O-ACETAL LEVULINYL ESTER GROUPS AND THEIR USE IN RNA MICROARRAYS WISCONSIN ALUMNI RESEARCH FOUNDATION (US) 2012-07-12 US claimed
EP-2334692-A1 RNA MONOMERS CONTAINING O-ACETAL LEVULINYL ESTER GROUPS AND THEIR USE IN RNA MICROARRAYS The Royal Institution for the Advancement of Learning / McGill University (CA) 2011-06-22 EP claimed
WO-2010025566-A1 RNA MONOMERS CONTAINING O-ACETAL LEVULINYL ESTER GROUPS AND THEIR USE IN RNA MICROARRAYS THE ROYAL INSTITUTION FOR THE ADVANCEMENT OF LEARNING/MCGILL UNIVERSITY (CA) 2010-03-11 WO claimed
EP-0934330-A1 BASE-PROTECTED NUCLEOTIDE ANALOGS WITH PROTECTED THIOL GROUPS Hanna, Michelle M. (US) 1999-08-11 EP claimed
WO-1998003532-A9 BASE-PROTECTED NUCLEOTIDE ANALOGS WITH PROTECTED THIOL GROUPS 1998-05-28 WO claimed
WO-1998003532-A1 BASE-PROTECTED NUCLEOTIDE ANALOGS WITH PROTECTED THIOL GROUPS HANNA MICHELLE M (US) 1998-01-29 WO claimed
WO-1994001445-A1 BASE-PROTECTED NUCLEOTIDE ANALOGS WITH PROTECTED THIOL GROUPS RESEARCH CORPORATION TECHNOLOGIES, INC. (US) 1994-01-20 WO claimed
WO-2026106497-A2 FUNCTIONALIZED CIRCULAR RNA AND METHODS AND INTERMEDIATES FOR THEIR PRODUCTION SIEĆ BADAWCZA ŁUKASIEWICZ – PORT POLSKI OSRODEK ROZWOJU TECHNOLOGII (PL) 2026-05-21 WO disclosed
WO-2025060642-A1 MODIFIED NUCLEOTIDE COMPOUND, OLIGONUCLEOTIDE THEREOF, AND USE THEREOF 广州必贝特医药股份有限公司 2025-03-27 WO disclosed
WO-1994019023-A1 CYCLOBUTYL ANTISENSE OLIGONUCLEOTIDES, METHODS OF MAKING AND USE THEREOF ISIS PHARMACEUTICALS, INC. (US) 1994-09-01 WO disclosed
WO-1994001445-A1 BASE-PROTECTED NUCLEOTIDE ANALOGS WITH PROTECTED THIOL GROUPS RESEARCH CORPORATION TECHNOLOGIES, INC. (US) 1994-01-20 WO disclosed
EP-0136693-A2 Production of cytidine derivatives Takeda Chemical Industries, Ltd. (JP) 1985-04-10 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10287313-B2 RNA monomers containing 0-acetal levulinyl ester groups and their use in RNA microarrays EFTUD2, RNMT, NSUN2 ADORA3 1812/4885ADORA1 2437/4885ADORA2A 1414/4885
US-11180756-B2 Morpholino modified oligomeric compounds RBM17, RBM3, UPF1 ADORA3 4054/4885ADORA1 4359/4885ADORA2A 4324/4885
US-20160340382-A1 RNA MONOMERS CONTAINING O-ACETAL LEVULINYL ESTER GROUPS AND THEIR USE IN RNA MICROARRAYS EFTUD2, RNMT, RNGTT ADORA3 1769/4885ADORA1 2519/4885ADORA2A 1438/4885
US-20200239881-A1 MORPHOLINO MODIFIED OLIGOMERIC COMPOUNDS RBM17, RBM3, UPF1 ADORA3 4054/4885ADORA1 4359/4885ADORA2A 4324/4885
US-20120178638-A1 RNA MONOMERS CONTAINING O-ACETAL LEVULINYL ESTER GROUPS AND THEIR USE IN RNA MICROARRAYS EFTUD2, RNMT, RNGTT ADORA3 1769/4885ADORA1 2519/4885ADORA2A 1438/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.