SCHEMBL21899482

SCHEMBL21899482

CNc1cnn2c(Cl)nc(-c3cncc(F)c3)nc12

nearest known ligand 0.35

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
AHR P35869 1/20 0.35
TLR7 Q9NYK1 7/20 0.32
CYP11B2 P19099 8/20 0.32
CYP11B1 P15538 7/20 0.32
CYP17A1 P05093 2/20 0.32
KAT2B Q92831 1/20 0.32
BRD9 Q9H8M2 1/20 0.32
CYP3A4 P08684 1/20 0.32
NQO2 P16083 1/20 0.31
ADORA2B P29275 1/20 0.31
IDH1 O75874 1/20 0.30
ABL1 P00519 1/20 0.30
CYP19A1 P11511 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20542084 0.83 CYP11B2 (0.36) AHRTLR7CYP11B2CYP11B1CYP17A1
SCHEMBL21855471 0.81 AHR (0.35) AHRCYP11B2CYP11B1CYP17A1CYP3A4
SCHEMBL21754340 0.81 CDK2 (0.35) AHRTLR7CYP11B2CYP11B1CYP17A1
SCHEMBL20557664 0.80 AHR (0.33) AHRTLR7CYP11B2CYP11B1CYP17A1
SCHEMBL20541825 0.80 AHR (0.49) AHRTLR7CYP11B2CYP11B1CYP17A1
SCHEMBL20557924 0.80 CYP11B2 (0.34) AHRTLR7CYP11B2CYP11B1CYP17A1
SCHEMBL29619215 0.80 AHR (0.49) AHRTLR7CYP11B2CYP11B1CYP17A1
SCHEMBL22566871 0.78 CYP11B2 (0.34) AHRTLR7CYP11B2CYP11B1CYP17A1
SCHEMBL24408393 0.76 AHR (0.40) AHRTLR7CYP11B2CYP11B1IDH1
SCHEMBL21855494 0.76 HRH4 (0.39) AHRTLR7CYP11B2CYP11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020081636-A1 INDOLE AHR INHIBITORS AND USES THEREOF Ikena Oncology, Inc. (US) 2020-04-23 WO disclosed