SCHEMBL21901276

SCHEMBL21901276

COC(=O)CC/C=C/c1cccc(Br)c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A19 Q695T7 1/20 0.51
HSD17B3 P37058 1/20 0.50
CYP4F2 P78329 1/20 0.48
CYP4A11 Q02928 1/20 0.48
BACE1 P56817 1/20 0.48
AKT1 P31749 1/20 0.47
PKM P14618 1/20 0.46
MAOB P27338 3/20 0.45
MAOA P21397 2/20 0.45
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44
ALDH1A1 P00352 2/20 0.43
MAPT P10636 1/20 0.43
HTT P42858 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
POLB P06746 2/20 0.43
KDM4E B2RXH2 1/20 0.42
MAPK1 P28482 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10696920 0.92 SLC6A19 (0.49) SLC6A19HSD17B3CYP4F2CYP4A11BACE1
SCHEMBL21791369 0.82 HSD17B3 (0.56) SLC6A19HSD17B3BACE1PKMMAOB
SCHEMBL19599777 0.82 HPGD (0.50) CYP4F2CYP4A11AKT1MAOBMAOA
SCHEMBL571591 0.82 HSD17B3 (0.56) SLC6A19HSD17B3BACE1PKMMAOB
SCHEMBL571592 0.82 HSD17B3 (0.56) SLC6A19HSD17B3BACE1PKMMAOB
SCHEMBL19452350 0.82 AKT1 (0.62) CYP4F2CYP4A11AKT1MAOBMEN1
SCHEMBL7571411 0.82 AKT1 (0.62) CYP4F2CYP4A11AKT1MAOBMEN1
SCHEMBL10698275 0.80 P4HB (0.51) CYP4F2CYP4A11AKT1MAOBMAOA
SCHEMBL10698280 0.80 P4HB (0.51) CYP4F2CYP4A11AKT1MAOBMAOA
SCHEMBL10699103 0.79 SLC6A19 (0.47) SLC6A19HSD17B3CYP4F2CYP4A11BACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2704571-B1 AMINO-PYRIDINE-CONTAINING SPLEEN TYROSINE KINASE (SYK) INHIBITORS MERCK SHARP & DOHME (US) 2020-04-22 EP disclosed