SCHEMBL21901752

SCHEMBL21901752

C=Cc1ccc(CC(C)(CO)CO)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.42
THRB P10828 2/20 0.40
THRA P10827 1/20 0.40
CYP3A4 P08684 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
ESR1 P03372 4/20 0.36
TDP1 Q9NUW8 1/20 0.34
ESR2 Q92731 3/20 0.33
TSHR P16473 1/20 0.33
HDAC8 Q9BY41 1/20 0.33
TAS1R3 Q7RTX0 1/20 0.32
TAS1R1 Q7RTX1 1/20 0.32
CHRNA4 P43681 2/20 0.31
CHRNB2 P17787 1/20 0.31
CHRNB4 P30926 1/20 0.31
CHRNA3 P32297 1/20 0.31
CHRNA7 P36544 1/20 0.31
TRPA1 O75762 2/20 0.31
TNNC1 P63316 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21901755 0.85 THRA (0.36) ALDH1A1THRBTHRACYP3A4CYP2C9
SCHEMBL21330385 0.80 ALDH1A1 (0.46) ALDH1A1THRBTHRACYP3A4CYP2C9
SCHEMBL1611980 0.79 THRA (0.53) ALDH1A1THRBTHRACYP3A4CYP2C9
SCHEMBL27520515 0.76 SLC6A2 (0.55) ALDH1A1THRBTHRAESR1TDP1
SCHEMBL10597489 0.76 ALDH1A1 (0.46) ALDH1A1THRBTHRACYP3A4CYP2C9
SCHEMBL5199704 0.74 ALDH1A1 (0.44) ALDH1A1THRBTHRACYP3A4CYP2C9
SCHEMBL6289217 0.74 ALDH1A1 (0.44) ALDH1A1THRBTHRACYP3A4CYP2C9
SCHEMBL14652352 0.74 ALDH1A1 (0.39) ALDH1A1THRBTHRACYP3A4CYP2C9
SCHEMBL9332631 0.74 THRA (0.41) ALDH1A1THRBTHRACYP3A4CYP2C9
SCHEMBL14268192 0.73 ALDH1A1 (0.42) ALDH1A1THRBTHRACYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20210189021-A1 CATALYST COMPOSITION, METHOD FOR PRODUCING MODIFIED CONJUGATED DIENE-BASED POLYMER, MODIFIED CONJUGATED DIENE-BASED POLYMER, RUBBER COMPOSITION, AND TIRE BRIDGESTONE CORPORATION (JP) 2021-06-24 US disclosed
EP-3640266-A1 CATALYST COMPOSITION, PRODUCTION METHOD FOR MODIFIED CONJUGATED DIENE POLYMER, MODIFIED CONJUGATED DIENE POLYMER, RUBBER COMPOSITION, AND TIRE Bridgestone Corporation (JP) 2020-04-22 EP disclosed