SCHEMBL21902913

SCHEMBL21902913

CC(C)CCc1ccc(CC(C)C)c(F)c1

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 2/20 0.41
GABRB2 P47870 2/20 0.41
RORC P51449 1/20 0.34
DPP4 P27487 2/20 0.33
ESR1 P03372 1/20 0.33
ALDH1A1 P00352 1/20 0.33
MAPT P10636 1/20 0.33
HTT P42858 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
GRIN2D O15399 1/20 0.33
GRIN2A Q12879 1/20 0.33
GRIN2B Q13224 1/20 0.33
GRIN2C Q14957 1/20 0.33
KCNH2 Q12809 2/20 0.32
TMEM97 Q5BJF2 2/20 0.32
SIGMAR1 Q99720 2/20 0.32
P2RX3 P56373 3/20 0.32
S1PR1 P21453 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21902910 0.86 GABRA1 (0.44) GABRA1GABRB2DPP4ALDH1A1MAPT
SCHEMBL12413798 0.86 GABRA1 (0.41) GABRA1GABRB2RORCDPP4SIGMAR1
SCHEMBL11809009 0.85 GABRA1 (0.55) GABRA1GABRB2RORCDPP4ESR1
SCHEMBL24233039 0.81 GABRA1 (0.43) GABRA1GABRB2RORCDPP4ALDH1A1
SCHEMBL12436729 0.81 ALDH1A1 (0.45) DPP4ALDH1A1MAPTHTTL3MBTL1
SCHEMBL9389779 0.80 BCHE (0.47) GABRA1GABRB2RORCS1PR1
SCHEMBL9389759 0.80 GABRA1 (0.46) GABRA1GABRB2RORCDPP4ESR1
SCHEMBL9390909 0.79 BCHE (0.49) GABRA1GABRB2S1PR1
SCHEMBL2741641 0.76 KDM4E (0.42) GABRA1GABRB2ESR1ALDH1A1MAPT
SCHEMBL12413796 0.75 GABRA1 (0.44) GABRA1GABRB2RORCMAPTS1PR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020078933-A1 PROTEOLYSIS TARGETING CHIMERA (PROTACS) AS DEGRADERS OF SMARCA2 AND/OR SMARCA4 BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2020-04-23 WO disclosed