SCHEMBL12413798

SCHEMBL12413798

CCCc1ccc(CC(C)C)c(F)c1

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 2/20 0.41
GABRB2 P47870 2/20 0.41
CNR1 P21554 1/20 0.39
CNR2 P34972 1/20 0.39
RORC P51449 1/20 0.37
PPARG P37231 1/20 0.35
PPARA Q07869 1/20 0.35
ALOX5 P09917 1/20 0.35
NPC1 O15118 1/20 0.34
TP53 P04637 1/20 0.34
PKM P14618 1/20 0.34
RAB9A P51151 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
HSD17B10 Q99714 1/20 0.34
DPP4 P27487 2/20 0.33
SIGMAR1 Q99720 1/20 0.33
S1PR1 P21453 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13003907 0.86 CNR1 (0.37) CNR1CNR2ALOX5NPC1TP53
SCHEMBL12413796 0.86 GABRA1 (0.44) GABRA1GABRB2RORCPPARGPPARA
SCHEMBL21902913 0.86 GABRA1 (0.41) GABRA1GABRB2RORCDPP4SIGMAR1
SCHEMBL24233039 0.85 GABRA1 (0.43) GABRA1GABRB2RORCNPC1RAB9A
SCHEMBL11809009 0.85 GABRA1 (0.55) GABRA1GABRB2RORCALOX5DPP4
SCHEMBL5165465 0.82 GABRA1 (0.53) GABRA1GABRB2CNR1CNR2PPARG
SCHEMBL15495007 0.81 CNR1 (0.44) CNR1CNR2ALOX5NPC1TP53
SCHEMBL9389779 0.80 BCHE (0.47) GABRA1GABRB2RORCS1PR1
SCHEMBL9389759 0.80 GABRA1 (0.46) GABRA1GABRB2RORCALOX5DPP4
SCHEMBL9390909 0.79 BCHE (0.49) GABRA1GABRB2S1PR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8293729-B2 Compounds, pharmaceutical composition and methods relating thereto BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2012-10-23 US disclosed
US-8293729-B2 Compounds, pharmaceutical composition and methods relating thereto BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2012-10-23 US disclosed
US-20110166116-A1 NEW COMPOUNDS, PHARMACEUTICAL COMPOSITION AND METHODS RELATING THERETO BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2011-07-07 US disclosed
US-20110166116-A1 NEW COMPOUNDS, PHARMACEUTICAL COMPOSITION AND METHODS RELATING THERETO BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2011-07-07 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110166116-A1 NEW COMPOUNDS, PHARMACEUTICAL COMPOSITION AND METHODS RELATING THERETO MC2R, REN, CYP11B2 GABRA1 1921/4885GABRB2 2941/4885CNR1 65/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.