Morpholine

Morpholine

SCHEMBL219044

C1COCCN1.CC(=O)O

nearest known ligand 0.58

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ADRA2AADRA2BADRA2CADRB2AGTR1AVPR1AAVPR1BAVPR2BDKRB2CALCRCHRNA3CHRNB4ESR1ESR2GHSRGNRHRGSC1HSPA8MALT1MC1RMC4RNOS1NOS2NOS3OPRK1OXTRRAMP1RAMP2RAMP3SCN5ASSTR1SSTR2SSTR3SSTR4SSTR5dacAdacBdacCfolPftsImrcAmrcBmrdArplArplBrplCrplDrplErplFrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmFrpmGrpmHrpmIrpmJrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of Morpholine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.58
MEN1 O00255 1/20 0.58
KDM4E B2RXH2 1/20 0.58
GAA P10253 1/20 0.58
CYP2C9 P11712 1/20 0.58
FFAR3 O14843 1/20 0.39
LCK P06239 1/20 0.39
FYN P06241 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.37
GABRP O00591 1/20 0.35
GABRD O14764 1/20 0.35
GABRA1 P14867 1/20 0.35
TSHR P16473 1/20 0.35
GABRB1 P18505 1/20 0.35
GABRG2 P18507 1/20 0.35
GABRB3 P28472 1/20 0.35
GABRA5 P31644 1/20 0.35
GABRA3 P34903 1/20 0.35
GABRA2 P47869 1/20 0.35
GABRB2 P47870 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Morpholine SCHEMBL29207396 1.00 KMT2A (0.58) KMT2AMEN1KDM4EGAACYP2C9
Acetic Acid SCHEMBL10708681 0.97 MEN1 (0.63) KMT2AMEN1KDM4EGAACYP2C9
Morpholine SCHEMBL29076892 0.97 KMT2A (0.55) KMT2AMEN1KDM4EGAACYP2C9
Acetic Acid SCHEMBL10707147 0.97 MEN1 (0.63) KMT2AMEN1KDM4EGAACYP2C9
Acetic Acid SCHEMBL28048691 0.97 KDM4E (0.63) KMT2AMEN1KDM4EGAACYP2C9
Morpholine SCHEMBL15572639 0.95 MEN1 (0.52) KMT2AMEN1KDM4EGAACYP2C9
Morpholine SCHEMBL15572290 0.95 MEN1 (0.52) KMT2AMEN1KDM4EGAACYP2C9
Morpholine SCHEMBL27737341 0.92 GAA (0.61) KMT2AMEN1KDM4EGAACYP2C9
Morpholine SCHEMBL15510851 0.91 MEN1 (0.48) KMT2AMEN1KDM4EGAACYP2C9
Morpholine SCHEMBL28632200 0.91 KMT2A (0.48) KMT2AMEN1KDM4EGAACYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 440 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110964085-B Preparation method of carfilzomib and derivatives thereof 扬子江药业集团有限公司 2023-07-07 CN claimed
CN-114524721-A Synthesis process of methacrolein 郑州中科新兴产业技术研究院 2022-05-24 CN claimed
CN-113786711-A Method for recovering chlorine-containing volatile organic compounds in organic waste gas by using ionic liquid 郑州中科新兴产业技术研究院 2021-12-14 CN claimed
US-10464958-B2 Method for the synthesis of alpha-aminoalkylenephosphonic acid MONSANTO TECHNOLOGY LLC (US) 2019-11-05 US claimed
CN-108997463-A A kind of female steroid -4,9- diene -3,17- diketone preparation method 四川理工学院 2018-12-14 CN claimed
US-20180346497-A1 METHOD FOR THE SYNTHESIS OF ALPHA-AMINOALKYLENEPHOSPHONIC ACID MONSANTO TECHNOLOGY LLC (US) 2018-12-06 US claimed
CN-103205000-B The preparation and application of ionic liquid 粟维清 2018-06-01 CN claimed
EP-3101026-B1 COMPOUNDS FOR PROTEASOME ENZYME INHIBITION ONYX THERAPEUTICS INC (US) 2018-03-28 EP claimed
EP-3101026-A1 COMPOUNDS FOR PROTEASOME ENZYME INHIBITION Onyx Therapeutics, Inc. (US) 2016-12-07 EP claimed
US-20150232493-A1 METHOD FOR THE SYNTHESIS OF ALPHA-AMINOALKYLENEPHOSPHONIC ACID MONSANTO TECHNOLOGY LLC 2015-08-20 US claimed
EP-1588145-A4 METHODS, MIXTURES, KITS AND COMPOSITIONS PERTAINING TO ANALYTE DETERMINATION APPLERA CORP (US) 2007-05-16 EP claimed
US-7195751-B2 Compositions and kits pertaining to analyte determination APPLERA CORPORATION (US) 2007-03-27 US claimed
CN-1762596-A Catalyst system for synthesizing acetic acid by methanol low-pressure carbonylation and its application SW RES & DESIGN INST CHEM IND (CN) 2006-04-26 CN claimed
CN-1740131-A Low pressure methanol carboxylating process to synthesize acetic acid SOUTHWEST CHEMICAL ENGINEERING (CN) 2006-03-01 CN claimed
EP-1588145-A2 METHODS, MIXTURES, KITS AND COMPOSITIONS PERTAINING TO ANALYTE DETERMINATION Applera Corporation (US) 2005-10-26 EP claimed
US-20040220412-A1 Compositions and kits pertaining to analyte determination APPLE CORPORATION 2004-11-04 US claimed
WO-2004070352-A2 METHODS, MIXTURES, KITS AND COMPOSITIONS PERTAINING TO ANALYTE DETERMINATION APPLERA CORPORATION (US) 2004-08-19 WO claimed
US-6028231-A Process for preparing 2-methyl-4-(2,2,3-trimethyl-cyclopent-3-en-1-yl)-but-2-en-1-ol HENKEL KOMMANDITGESELLSCHAFT AUF AKTIEN (DE) 2000-02-22 US claimed
WO-1999035219-A1 HYDRAULIC FLUIDS CONTAINING N-ALKYL MORPHOLINE OR A SALT THEREOF MACDERMID EUROPE PLC (GB) 1999-07-15 WO claimed
US-4298477-A Regeneration of cation ion-exchange polishers NALCO CHEMICAL COMPANY (US) 1981-11-03 US claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040220412-A1 Compositions and kits pertaining to analyte determination KLK3, SRMS, SHBG KMT2A 3232/4885MEN1 389/4885KDM4E 4358/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.