SCHEMBL21914701

SCHEMBL21914701

COc1cccc(CN2N=C(/C(C)=C/C=C(\C)Cl)c3ccsc3-n3c(C)nnc32)c1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.35
BRD4 O60885 1/20 0.34
P2RX7 Q99572 1/20 0.34
CYP2D6 P10635 3/20 0.33
CYP2C19 P33261 3/20 0.33
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
ALDH1A1 P00352 2/20 0.33
USP2 O75604 2/20 0.33
CYP1A2 P05177 2/20 0.33
CYP3A4 P08684 2/20 0.33
CYP2C9 P11712 2/20 0.33
LMNA P02545 1/20 0.33
TSHR P16473 1/20 0.33
CLK4 Q9HAZ1 1/20 0.33
SIGMAR1 Q99720 1/20 0.32
CLK1 P49759 1/20 0.32
DYRK1A Q13627 1/20 0.32
CD74 P04233 1/20 0.32
MIF P14174 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21847283 0.79 ALDH1A1 (0.39) BRD4P2RX7CYP2C19MEN1KMT2A
SCHEMBL21847192 0.68 BRD4 (0.39) SMN1; SMN2BRD4CYP2D6ALDH1A1USP2
SCHEMBL21847101 0.66 BRD4 (0.41) BRD4CYP2D6CYP2C19MEN1KMT2A
SCHEMBL21847138 0.66 BRD4 (0.46) BRD4
SCHEMBL21847285 0.65 BRD4 (0.43) SMN1; SMN2BRD4ALDH1A1USP2LMNA
SCHEMBL8319389 0.65 BRD4 (0.46) BRD4P2RX7CYP2D6LMNA
SCHEMBL21847118 0.62 P2RX7 (0.38) BRD4P2RX7
SCHEMBL21847113 0.61 BRD4 (0.37) BRD4ALDH1A1
SCHEMBL21847104 0.60 PDE4B (0.40) BRD4CYP2D6CYP2C19MEN1KMT2A
SCHEMBL21847182 0.59 BRD4 (0.41) SMN1; SMN2BRD4CYP2D6LMNATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3640253-A1 6H-THIENO[2,3-E][1,2,4]TRIAZOLO[3,4-C][1,2,4]TRIAZEPINE DERIVATIVE AYUMI Pharmaceutical Corporation (JP) 2020-04-22 EP disclosed