SCHEMBL21925264

SCHEMBL21925264

Cc1cccc(C2CCCN(F)C2)n1

nearest known ligand 0.49

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MAP4K4 O95819 2/20 0.49
KDM5A P29375 1/20 0.44
DRD2 P14416 9/20 0.40
DRD4 P21917 9/20 0.40
HTR1A P08908 8/20 0.40
CNR2 P34972 2/20 0.40
OPRM1 P35372 1/20 0.40
OPRL1 P41146 1/20 0.40
KCNH2 Q12809 3/20 0.38
CXCR4 P61073 1/20 0.37
PDE2A O00408 2/20 0.37
CCR1 P32246 1/20 0.36
CCR8 P51685 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12090447 0.83 MAP4K4 (0.50) MAP4K4KDM5ADRD2DRD4HTR1A
SCHEMBL23114442 0.83 MAP4K4 (0.50) MAP4K4KDM5ADRD2DRD4HTR1A
SCHEMBL17896370 0.82 DRD2 (0.49) MAP4K4KDM5ADRD2DRD4HTR1A
SCHEMBL2757250 0.78 CCR1 (0.48) MAP4K4DRD2DRD4HTR1ACNR2
SCHEMBL15087991 0.78 CCR1 (0.48) MAP4K4KDM5ADRD2DRD4HTR1A
SCHEMBL8056158 0.77 DRD2 (0.50) MAP4K4DRD2DRD4HTR1ACNR2
SCHEMBL171619 0.76 PDE2A (0.55) MAP4K4DRD2DRD4KCNH2PDE2A
SCHEMBL1610517 0.74 CCR1 (0.52) MAP4K4KDM5ADRD2DRD4HTR1A
SCHEMBL20139964 0.74 KDM5A (0.58) MAP4K4KDM5ADRD2DRD4HTR1A
SCHEMBL17888476 0.72 DRD2 (0.53) MAP4K4KDM5ADRD2DRD4HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2855459-B1 AMINOQUINAZOLINE AND PYRIDOPYRIMIDINE DERIVATIVES HOFFMANN LA ROCHE (CH) 2020-04-29 EP disclosed