SCHEMBL20139964

SCHEMBL20139964

Cc1cccc([C@H]2CCN(C(=O)O)C2)n1

nearest known ligand 0.58

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
KDM5A P29375 5/20 0.58
DRD2 P14416 10/20 0.49
DRD4 P21917 10/20 0.49
HTR1A P08908 9/20 0.49
KCNH2 Q12809 4/20 0.46
MAP4K4 O95819 1/20 0.42
PDE10A Q9Y233 1/20 0.42
MAP3K12 Q12852 1/20 0.42
CNR2 P34972 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20139993 0.91 DRD2 (0.54) KDM5ADRD2DRD4HTR1AKCNH2
SCHEMBL1740301 0.88 KDM5A (0.48) KDM5ADRD2DRD4HTR1AKCNH2
SCHEMBL20140687 0.82 KDM5A (0.53) KDM5ADRD2DRD4HTR1AKCNH2
SCHEMBL20157283 0.82 KDM5A (0.53) KDM5ADRD2DRD4HTR1AKCNH2
SCHEMBL17672417 0.79 KDM5A (0.47) KDM5A
SCHEMBL2806341 0.77 HSD11B1 (0.60) KDM5ADRD2DRD4
SCHEMBL20140593 0.76 HTR1A (0.54) DRD2DRD4HTR1AKCNH2
SCHEMBL27727712 0.76 KDM4E (0.53) KDM5AMAP4K4MAP3K12
SCHEMBL17820444 0.75 PDE10A (0.43) KDM5APDE10ACNR2
SCHEMBL17682618 0.75 KDM5A (0.69) KDM5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018089433-A1 PHENYL mTORC INHIBITORS AND USES THEREOF NAVITOR PHARMACEUTICALS, INC. (US) 2018-05-17 WO disclosed