SCHEMBL21936050

SCHEMBL21936050

Cc1c(C=O)nc2cc(Br)ccn12

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.38
MAPT P10636 3/20 0.38
NPC1 O15118 2/20 0.38
RAB9A P51151 2/20 0.38
ALDH1A1 P00352 6/20 0.35
CYP11B1 P15538 2/20 0.35
CYP11B2 P19099 2/20 0.35
AHR P35869 2/20 0.33
AKT2 P31751 1/20 0.33
POLB P06746 2/20 0.33
RECQL P46063 1/20 0.33
MEN1 O00255 1/20 0.31
LMNA P02545 1/20 0.31
KMT2A Q03164 1/20 0.31
GAA P10253 2/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
CASP3 P42574 1/20 0.31
TP53 P04637 1/20 0.30
THRB P10828 1/20 0.30
GLA P06280 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23726410 0.81 ALDH1A1 (0.33) KDM4EMAPTALDH1A1AHRAKT2
SCHEMBL21937177 0.80 AHR (0.31) AHR
SCHEMBL21936037 0.80 HDAC1 (0.34) MAPTAHRPOLBRECQL
SCHEMBL974116 0.78 KDM4E (0.40) KDM4EMAPTNPC1RAB9AALDH1A1
SCHEMBL31528577 0.76 RAB9A (0.49) KDM4EMAPTNPC1RAB9AALDH1A1
SCHEMBL870880 0.75 ALDH1A1 (0.55) KDM4EMAPTNPC1RAB9AALDH1A1
SCHEMBL23726594 0.74 MAPT (0.41) KDM4EMAPTNPC1RAB9AALDH1A1
SCHEMBL25327960 0.73 ALDH1A1 (0.41) KDM4EMAPTNPC1RAB9AALDH1A1
SCHEMBL15766770 0.71 KDM4E (0.38) KDM4EMAPTNPC1RAB9AALDH1A1
SCHEMBL24798078 0.71 CYP2A6 (0.36) KDM4EMAPTNPC1RAB9AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112601745-B Azaaryl amide derivative and preparation method and application thereof 上海和誉生物医药科技有限公司 2023-06-27 CN disclosed
CN-112601745-A Azaaryl amide derivative and preparation method and application thereof 上海和誉生物医药科技有限公司 2021-04-02 CN disclosed
WO-2020082921-A1 NITROGEN HETEROARYL AMIDE DERIVATIVE, PREPARATION METHOD THEREFOR, AND APPLICATION THEREOF 上海和誉生物医药科技有限公司 2020-04-30 WO disclosed