SCHEMBL2194496

SCHEMBL2194496

O=C(c1ccc(Br)cc1)N(Cc1ccccc1)c1cccnc1

nearest known ligand 0.70

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.70
GAA P10253 2/20 0.70
CHRM3 P20309 1/20 0.56
KMT2A Q03164 4/20 0.52
NPC1 O15118 2/20 0.52
MEN1 O00255 2/20 0.52
HTT P42858 1/20 0.50
STAT3 P40763 1/20 0.47
RAB9A P51151 1/20 0.46
PDK1 Q15118 2/20 0.45
NR1H4 Q96RI1 1/20 0.44
TRPV1 Q8NER1 1/20 0.44
LTB4R2 Q9NPC1 1/20 0.43
CYP11B1 P15538 1/20 0.43
CYP11B2 P19099 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13571398 0.91 TSHR (0.84) TSHRGAAKMT2ANPC1MEN1
SCHEMBL28807373 0.83 GAA (0.70) TSHRGAAKMT2ANPC1HTT
SCHEMBL2194451 0.79 TSHR (0.69) TSHRGAAKMT2AMEN1HTT
SCHEMBL3060251 0.78 TSHR (0.71) TSHRGAAKMT2ANPC1MEN1
SCHEMBL22289326 0.76 GAA (0.73) TSHRGAAKMT2ANPC1HTT
SCHEMBL1336782 0.76 GAA (0.60) TSHRGAAKMT2ANPC1HTT
SCHEMBL8332050 0.75 KMT2A (0.71) TSHRGAAKMT2ANPC1MEN1
SCHEMBL5907003 0.74 ALDH1A1 (0.54) TSHRGAACHRM3NPC1HTT
SCHEMBL14908642 0.72 SMN1; SMN2 (0.49) TSHRGAANPC1HTTRAB9A
SCHEMBL14720449 0.72 CHRM3 (0.52) TSHRGAACHRM3KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2519522-A2 SUBSTITUTED IMIDAZOPYRIDINYL-AMINOPYRIDINE COMPOUNDS ArQule, Inc. (US) 2012-11-07 EP disclosed
WO-2011082270-A2 SUBSTITUTED IMIDAZOPYRIDINYL-AMINOPYRIDINE COMPOUNDS ARQULE. INC. (US) 2011-07-07 WO disclosed