SCHEMBL14720449

SCHEMBL14720449

O=C(O)N1CC[C@@H](CN(C(=O)c2ccc(Br)cc2)c2cccnc2)C1

nearest known ligand 0.52

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CHRM3 P20309 2/20 0.52
CHRM2 P08172 1/20 0.39
CYP3A4 P08684 5/20 0.39
ACHE P22303 2/20 0.39
HTT P42858 1/20 0.38
VNN1 O95497 1/20 0.38
GAA P10253 1/20 0.38
TSHR P16473 1/20 0.38
CHRNB2 P17787 1/20 0.38
CHRNA7 P36544 1/20 0.38
CHRNA4 P43681 1/20 0.38
CYP2D6 P10635 1/20 0.37
CYP2C9 P11712 1/20 0.37
GRIN2B Q13224 1/20 0.37
ALDH1A1 P00352 1/20 0.36
MEN1 O00255 1/20 0.36
LMNA P02545 1/20 0.36
MAPK1 P28482 1/20 0.36
KMT2A Q03164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14720407 0.85 CHRM3 (0.39) CHRM3CHRM2CYP3A4ACHEVNN1
SCHEMBL14720297 0.76 LIMK2 (0.48) CHRM3CHRM2ACHEMEN1KMT2A
SCHEMBL14720201 0.75 HDAC1 (0.52) CHRM3CHRM2KMT2A
SCHEMBL14720757 0.74 CHRM3 (0.44) CHRM3CHRM2CYP3A4ACHEHTT
SCHEMBL14720344 0.74 OPRM1 (0.42) ALDH1A1
SCHEMBL14731351 0.74 FASN (0.50) CYP3A4
SCHEMBL14720668 0.73 OPRD1 (0.39) CHRM3CHRM2KMT2A
SCHEMBL14731350 0.73 FASN (0.57)
SCHEMBL2194496 0.72 TSHR (0.70) CHRM3HTTGAATSHRMEN1
SCHEMBL14720234 0.69 GRIN2B (0.64) CYP3A4VNN1CYP2D6CYP2C9GRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013028445-A1 FATTY ACID SYNTHASE INHIBITORS GLAXOSMITHKLINE LLC (US) 2013-02-28 WO disclosed