SCHEMBL21963465

SCHEMBL21963465

O=c1[nH]ccc2sc(-c3ccc(Cl)cc3)cc12

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 4/20 0.40
LMNA P02545 2/20 0.40
KDM4E B2RXH2 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
CYP1A1 P04798 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP1B1 Q16678 1/20 0.40
CHEK1 O14757 1/20 0.40
ALDH1A1 P00352 6/20 0.39
HPGD P15428 2/20 0.39
PTP4A3 O75365 1/20 0.38
PTP4A2 Q12974 1/20 0.38
PTP4A1 Q93096 1/20 0.38
PARP1 P09874 2/20 0.38
IKBKB O14920 1/20 0.38
MAPT P10636 3/20 0.37
POLB P06746 1/20 0.37
GSK3B P49841 3/20 0.37
PRKDC P78527 1/20 0.36
NPC1 O15118 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4515919 0.84 RAB9A (0.55) RAB9ALMNAKDM4ESMN1; SMN2ALDH1A1
SCHEMBL14911794 0.81 GSK3B (0.56) RAB9ALMNAALDH1A1HPGDMAPT
SCHEMBL386804 0.75 RAB9A (0.49) RAB9ALMNAKDM4ESMN1; SMN2CYP1A1
SCHEMBL21963437 0.74 ELANE (0.42) RAB9ASMN1; SMN2ALDH1A1HPGDMAPT
SCHEMBL7835046 0.71 PARP1 (0.39) RAB9ALMNAKDM4ECYP1A2CHEK1
SCHEMBL1774094 0.69 PARP1 (0.43) RAB9ALMNAKDM4ECYP1A2CHEK1
SCHEMBL4341520 0.69 ALDH1A1 (0.47) RAB9ALMNAKDM4ECYP1A2CHEK1
SCHEMBL6226394 0.69 CHEK1 (0.50) CHEK1ALDH1A1PARP1IKBKB
SCHEMBL15716637 0.67 CYP2A6 (0.42) RAB9ALMNAKDM4ECYP1A2CHEK1
SCHEMBL5849531 0.66 TMIGD3 (0.51) RAB9ALMNAKDM4ESMN1; SMN2CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3880200-A2 IN-FLOW PHOTOOXYGENATION OF AMINOTHIENOPYRIDINONES GENERATES NOVEL PTP4A3 PHOSPHATASE INHIBITORS University of Virginia Patent Foundation (US) 2021-09-22 EP disclosed
EP-3880684-A1 IN-FLOW PHOTOOXYGENATION OF AMINOTHIENOPYRIDINONES GENERATES NOVEL PTP4A3 PHOSPHATASE INHIBITORS University of Virginia Patent Foundation (US) 2021-09-22 EP disclosed
WO-2020102243-A2 IN-FLOW PHOTOOXYGENATION OF AMINOTHIENOPYRIDINONES GENERATES NOVEL PTP4A3 PHOSPHATASE INHIBITORS UNIVERSITY OF VIRGINIA PATENT FOUNDATION (US) 2020-05-22 WO disclosed
WO-2020102245-A1 IN-FLOW PHOTOOXYGENATION OF AMINOTHIENOPYRIDINONES GENERATES NOVEL PTP4A3 PHOSPHATASE INHIBITORS UNIVERSITY OF VIRGINIA PATENT FOUNDATION (US) 2020-05-22 WO disclosed