SCHEMBL21972969

SCHEMBL21972969

CC1(N)C=CC=C(c2nc(-c3ccccc3)nc(-c3ccccc3)n2)C=C1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 2/20 0.41
ADORA2A P29274 5/20 0.37
ADORA1 P30542 4/20 0.37
ADORA3 P0DMS8 3/20 0.37
ADORA2B P29275 2/20 0.37
POLB P06746 1/20 0.37
KMT2A Q03164 7/20 0.36
MEN1 O00255 6/20 0.36
MAPT P10636 3/20 0.36
HPGD P15428 3/20 0.36
ALDH1A1 P00352 2/20 0.36
HTT P42858 1/20 0.34
NOTUM Q6P988 1/20 0.33
HSP90AA1 P07900 1/20 0.33
HSP90AB1 P08238 1/20 0.33
ALOX15 P16050 1/20 0.33
TSHR P16473 1/20 0.33
LMNA P02545 3/20 0.32
KDM4E B2RXH2 3/20 0.32
ATM Q13315 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20829144 0.90 RAB9A (0.43) L3MBTL1ADORA1KMT2AMEN1MAPT
SCHEMBL20829145 0.88 ADORA2A (0.41) L3MBTL1ADORA2AADORA1KMT2AMEN1
SCHEMBL20829147 0.86 MEN1 (0.45) L3MBTL1ADORA2AADORA1ADORA3KMT2A
SCHEMBL21233511 0.85 KDM1A (0.31)
SCHEMBL25923595 0.84 L3MBTL1 (0.43) L3MBTL1ADORA2AADORA1ADORA3ADORA2B
SCHEMBL26730292 0.83 L3MBTL1 (0.42) L3MBTL1ADORA2AADORA1ADORA3ADORA2B
SCHEMBL22296632 0.79 L3MBTL1 (0.54) L3MBTL1ADORA2AADORA1ADORA3ADORA2B
SCHEMBL20829146 0.79 ADORA2A (0.38) L3MBTL1ADORA2AADORA1POLBKMT2A
SCHEMBL21973501 0.78 IKBKB (0.33)
SCHEMBL20829149 0.77 MEN1 (0.40) L3MBTL1ADORA2AADORA1ADORA3ADORA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3423542-B1 MATERIALS FOR ORGANIC ELECTROLUMINESCENT DEVICES MERCK PATENT GMBH (DE) 2020-07-22 EP disclosed
EP-3197982-B1 MATERIALS FOR ORGANIC ELECTROLUMINESCENT DEVICES MERCK PATENT GMBH (DE) 2020-05-06 EP disclosed