SCHEMBL21974992

SCHEMBL21974992

CNc1nc(-c2cccnc2)nc(Oc2cc(C(=O)Nc3cc(C(F)(F)F)cc(C(F)(F)F)c3)ccc2C)c1C=N

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 7/20 0.49
TEK Q02763 6/20 0.49
YES1 P07947 4/20 0.49
ABL1 P00519 10/20 0.48
BCR P11274 7/20 0.48
RET P07949 4/20 0.48
MAPK14 Q16539 4/20 0.48
EPHB6 O15197 3/20 0.48
STK10 O94804 3/20 0.48
LCK P06239 3/20 0.48
FYN P06241 3/20 0.48
LYN P07948 3/20 0.48
HCK P08631 3/20 0.48
PDGFRB P09619 3/20 0.48
SRC P12931 3/20 0.48
BRAF P15056 3/20 0.48
PHKG2 P15735 3/20 0.48
NQO2 P16083 3/20 0.48
EPHA1 P21709 3/20 0.48
FECH P22830 3/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21975658 0.94 KDR (0.57) KDRTEKYES1ABL1BCR
SCHEMBL21975688 0.89 ABL1 (0.45) KDRTEKYES1ABL1BCR
SCHEMBL21975119 0.82 RET (0.39) RETBRAFLMNAHSD17B10KIF5B
SCHEMBL21943600 0.80 ABL1 (0.67) KDRTEKYES1ABL1BCR
SCHEMBL21974774 0.80 RET (0.71) ABL1BCRRETLCKLYN
SCHEMBL22066074 0.78 BRAF (0.61) KDRTEKYES1ABL1BCR
SCHEMBL21975103 0.77 CYP1A2 (0.41) PRKCAMAPK1RECQLHSD17B10CLK4
SCHEMBL21975693 0.77 LRRK2 (0.44) TTK
SCHEMBL21975115 0.76 POLB (0.48) RETLMNADYRK1AKIF5BCCDC6
SCHEMBL21975647 0.73 ABCG2 (0.48) KDRTEKYES1MAPK14PDGFRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3647313-A1 SUBSTITUTED ARYL ETHER COMPOUND, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION AND USE THEREOF Xiamen University (CN) 2020-05-06 EP disclosed