SCHEMBL22066074

SCHEMBL22066074

CNc1nc(-c2cccnc2)nc(Nc2cc(NC(=O)c3cccc(C(F)(F)F)c3)ccc2C)c1C=N

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRAF P15056 10/20 0.61
CSF1R P07333 4/20 0.61
PIKFYVE Q9Y2I7 2/20 0.61
ABL1 P00519 4/20 0.60
BCR P11274 3/20 0.60
SRC P12931 3/20 0.60
DDR1 Q08345 3/20 0.60
MAPK14 Q16539 3/20 0.60
DDR2 Q16832 3/20 0.60
ESYT2 A0FGR8 2/20 0.60
NBAS A2RRP1 2/20 0.60
CNOT1 A5YKK6 2/20 0.60
TBKBP1 A7MCY6 2/20 0.60
AGPS O00116 2/20 0.60
MYO1F O00160 2/20 0.60
SNAP23 O00161 2/20 0.60
AP3B1 O00203 2/20 0.60
PSMD12 O00232 2/20 0.60
BMPR1B O00238 2/20 0.60
PGRMC1 O00264 2/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22066484 0.86 MAPK14 (0.68) BRAFCSF1RPIKFYVEABL1BCR
SCHEMBL22066412 0.85 POLB (0.57) BRAFCSF1RABL1BCRSRC
SCHEMBL22066322 0.83 LCK (0.54) BRAFCSF1RABL1BCRSRC
SCHEMBL21975658 0.83 KDR (0.57) BRAFCSF1RABL1BCRSRC
SCHEMBL22024838 0.82 PIKFYVE (0.80) BRAFCSF1RPIKFYVEABL1BCR
SCHEMBL22065355 0.82 LCK (0.54) BRAFCSF1RABL1BCRSRC
SCHEMBL22065360 0.82 POLB (0.53) BRAFCSF1RABL1BCRSRC
SCHEMBL22024547 0.82 PIKFYVE (0.65) BRAFCSF1RPIKFYVEABL1BCR
SCHEMBL22024570 0.82 PIKFYVE (0.77) BRAFCSF1RPIKFYVEABL1BCR
SCHEMBL24532075 0.81 BRAF (0.89) BRAFCSF1RPIKFYVEABL1BCR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3663293-A1 SUBSTITUTED PENTA- AND HEXA-HETEROCYCLIC COMPOUNDS, PREPARATION METHOD THEREFOR, DRUG COMBINATION AND USE THEREOF Xiamen University (CN) 2020-06-10 EP disclosed