SCHEMBL21976307

SCHEMBL21976307

CCOCCOc1ccccc1C1Nc2ccc(C(=O)NO)cc2N1

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 4/20 0.41
HDAC8 Q9BY41 4/20 0.41
HDAC6 Q9UBN7 4/20 0.41
LMNA P02545 2/20 0.41
ALDH1A1 P00352 2/20 0.41
SMPD1 P17405 8/20 0.40
TSHR P16473 1/20 0.40
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
TAAR1 Q96RJ0 1/20 0.39
DRD2 P14416 2/20 0.37
DRD4 P21917 2/20 0.37
DRD3 P35462 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21976490 0.92 SMN1; SMN2 (0.40) HDAC1HDAC8HDAC6LMNAALDH1A1
SCHEMBL21976232 0.90 SMPD1 (0.45) HDAC1HDAC8HDAC6ALDH1A1SMPD1
SCHEMBL21976248 0.87 HDAC6 (0.45) HDAC8HDAC6LMNAALDH1A1SMPD1
SCHEMBL21976229 0.75 GAA (0.46) HDAC1HDAC8HDAC6ALDH1A1TSHR
SCHEMBL21976306 0.73 HDAC6 (0.47) HDAC8HDAC6SMPD1MEN1KMT2A
SCHEMBL21976469 0.72 HDAC6 (0.47) HDAC1HDAC8HDAC6
SCHEMBL21976208 0.72 PBRM1 (0.44) HDAC1HDAC8HDAC6
SCHEMBL21975927 0.71 KDM4E (0.41) HDAC1HDAC8HDAC6SMPD1
SCHEMBL21976479 0.71 HDAC6 (0.50) HDAC1HDAC8HDAC6LMNASMPD1
SCHEMBL21976492 0.70 SMPD1 (0.53) HDAC6LMNAALDH1A1SMPD1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3294715-B1 BENZIMIDAZOLE DERIVATES USEFUL AS INHIBITORS OF MAMMALIAN HISTONE DEACETYLASE ACTIVITY KANCERA AB (SE) 2020-05-06 EP disclosed