SCHEMBL21976232

SCHEMBL21976232

CCCOc1ccccc1C1Nc2ccc(C(=O)NO)cc2N1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMPD1 P17405 8/20 0.45
HDAC1 Q13547 4/20 0.42
HDAC8 Q9BY41 3/20 0.42
HDAC6 Q9UBN7 3/20 0.42
GAA P10253 3/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
HDAC2 Q92769 1/20 0.41
ALDH1A1 P00352 2/20 0.40
HSD17B10 Q99714 2/20 0.40
MAPT P10636 1/20 0.40
ALOX15 P16050 1/20 0.40
KDM4E B2RXH2 1/20 0.40
GLA P06280 1/20 0.40
HPGD P15428 1/20 0.40
MAPK1 P28482 1/20 0.40
CASP1 P29466 1/20 0.40
CASP7 P55210 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
TP53 P04637 1/20 0.39
TSHR P16473 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21976307 0.90 HDAC1 (0.41) SMPD1HDAC1HDAC8HDAC6ALDH1A1
SCHEMBL21976490 0.88 SMN1; SMN2 (0.40) SMPD1HDAC1HDAC8HDAC6GAA
SCHEMBL21976248 0.88 HDAC6 (0.45) SMPD1HDAC8HDAC6ALDH1A1MAPT
SCHEMBL21976492 0.79 SMPD1 (0.53) SMPD1HDAC6SMN1; SMN2ALDH1A1MAPT
SCHEMBL21976229 0.77 GAA (0.46) HDAC1HDAC8HDAC6GAASMN1; SMN2
SCHEMBL21976208 0.74 PBRM1 (0.44) HDAC1HDAC8HDAC6KDM4E
SCHEMBL21976469 0.74 HDAC6 (0.47) HDAC1HDAC8HDAC6HDAC2KDM4E
SCHEMBL21975927 0.74 KDM4E (0.41) SMPD1HDAC1HDAC8HDAC6KDM4E
SCHEMBL21976306 0.73 HDAC6 (0.47) SMPD1HDAC8HDAC6MAPT
SCHEMBL21976478 0.72 ALOX5 (0.42) HDAC1HDAC8HDAC6GAAHDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3294715-B1 BENZIMIDAZOLE DERIVATES USEFUL AS INHIBITORS OF MAMMALIAN HISTONE DEACETYLASE ACTIVITY KANCERA AB (SE) 2020-05-06 EP disclosed