SCHEMBL21985307

SCHEMBL21985307

CN1CC(COc2c(Cl)cc(F)cc2Cl)C1

nearest known ligand 0.38

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 1/20 0.34
SLC5A1 P13866 1/20 0.34
SLC5A2 P31639 1/20 0.34
CHRM3 P20309 7/20 0.33
EPHA2 P29317 1/20 0.33
KDR P35968 1/20 0.33
EPHB4 P54760 1/20 0.33
MGLL Q99685 1/20 0.33
OPRL1 P41146 1/20 0.33
FFAR1 O14842 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7953445 0.86 HRH3 (0.43) CHRM3KDR
SCHEMBL21985038 0.80 MGLL (0.49) SLC6A4MGLL
Hydrochloric Acid SCHEMBL7954788 0.73 HRH3 (0.45) KDR
SCHEMBL17910956 0.73 LMNA (0.43)
SCHEMBL10267768 0.71 DRD4 (0.48)
SCHEMBL13416777 0.69 HSP90AA1 (0.42) KDR
Hydrochloric Acid SCHEMBL7953408 0.67 HRH3 (0.50) SLC6A4CHRM3
SCHEMBL20204779 0.66 MAPT (0.40) SLC6A4CHRM3KDRFFAR1
SCHEMBL13452598 0.66 MAOA (0.50) CHRM3KDR
SCHEMBL3841470 0.65 LMNA (0.40)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3436444-B1 HETEROCYCLIC COMPOUND TAKEDA PHARMACEUTICALS CO (JP) 2020-05-13 EP disclosed