SCHEMBL21986158

SCHEMBL21986158

Cc1cnc(I)c2occc12

nearest known ligand 0.35

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 1/20 0.32
CCR5 P51681 1/20 0.32
CCR8 P51685 1/20 0.32
DRD2 P14416 1/20 0.31
HTR2A P28223 1/20 0.31
DRD3 P35462 1/20 0.31
ASIC3 Q9UHC3 1/20 0.30
AXL P30530 1/20 0.30
PRKCI P41743 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8737213 0.80 CCR1 (0.34) CCR1CCR5CCR8DRD2HTR2A
SCHEMBL18820429 0.74 KCNA2 (0.33) CCR1CCR5CCR8DRD2HTR2A
SCHEMBL8737251 0.74 HTR2A (0.31) CCR1CCR5CCR8HTR2A
SCHEMBL8737765 0.74 CCR1 (0.35) CCR1CCR5CCR8DRD2HTR2A
SCHEMBL1698415 0.69 DRD2 (0.33) CCR1CCR5CCR8DRD2HTR2A
SCHEMBL30110578 0.69 DRD2 (0.33) CCR1CCR5CCR8DRD2HTR2A
SCHEMBL15688334 0.69 NOS2 (0.41) CCR1CCR5CCR8DRD2HTR2A
SCHEMBL10217310 0.69 CYP2A6 (0.31)
SCHEMBL31120928 0.68 CYP1A2 (0.39) CCR1CCR5CCR8HTR2A
SCHEMBL806473 0.68 CYP1A2 (0.39) CCR1CCR5CCR8HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3172214-B1 2-AMINO-PYRIDO[2,3-D]PYRIMIDIN-7(8H)-ONE DERIVATIVES AS CDK INHIBITORS AND USES THEREOF SUNSHINE LAKE PHARMA CO LTD (CN) 2020-05-13 EP disclosed