SCHEMBL21986361

SCHEMBL21986361

O=[C]N1CCN(c2cccc(Br)c2)c2ccccc21

nearest known ligand 0.46

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
BRD2 P25440 1/20 0.46
ALDH1A1 P00352 4/20 0.42
HSD11B1 P28845 1/20 0.40
MGLL Q99685 1/20 0.38
ALOX5 P09917 2/20 0.38
ATM Q13315 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
DHFR P00374 1/20 0.36
MEN1 O00255 4/20 0.35
KMT2A Q03164 4/20 0.35
POLB P06746 1/20 0.33
HTT P42858 1/20 0.33
CACNA2D1 P54289 1/20 0.33
TP53 P04637 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19280241 0.75 BRD2 (0.45) BRD2ALDH1A1HSD11B1MGLLALOX5
SCHEMBL14339392 0.73 ALDH1A1 (0.46) BRD2ALDH1A1HSD11B1MGLLALOX5
SCHEMBL28847051 0.70 MEN1 (0.53) BRD2ALDH1A1HSD11B1ALOX5L3MBTL1
SCHEMBL19280531 0.69 HDAC1 (0.45) BRD2ALDH1A1HSD11B1
SCHEMBL12543536 0.67 HSD11B1 (0.36) ALDH1A1HSD11B1MEN1KMT2A
SCHEMBL17870929 0.66 ALDH1A1 (0.54) ALDH1A1HSD11B1MGLLALOX5ATM
SCHEMBL18485726 0.65 BRD2 (0.61) BRD2ALDH1A1HSD11B1ALOX5DHFR
SCHEMBL21020694 0.65 ALDH1A1 (0.42) BRD2ALDH1A1HSD11B1MGLLALOX5
SCHEMBL18485728 0.64 BRD2 (0.54) BRD2ALDH1A1HSD11B1MGLLALOX5
SCHEMBL27574161 0.64 ALDH1A1 (0.41) ALDH1A1HSD11B1MGLLALOX5ATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3209664-B1 BICYCLIC HETEROARYL AMINE COMPOUNDS AS PI3K INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2020-06-03 EP disclosed