SCHEMBL2199143

SCHEMBL2199143

C[C@@H](c1ccc([C@H](O)CNC2(CO)CCCC2)cc1)N(C(=O)O)C(C)(C)C

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.38
BCHE P06276 1/20 0.34
KDM4E B2RXH2 4/20 0.32
ADRB2 P07550 4/20 0.32
BLM P54132 3/20 0.32
LMNA P02545 3/20 0.32
ADRB1 P08588 2/20 0.32
ADRB3 P13945 2/20 0.32
GLA P06280 1/20 0.32
POLB P06746 2/20 0.31
MAPT P10636 2/20 0.31
TDP1 Q9NUW8 2/20 0.31
MEN1 O00255 2/20 0.31
GAA P10253 1/20 0.31
RXFP1 Q9HBX9 1/20 0.31
TP53 P04637 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
ALOX15 P16050 1/20 0.31
TSHR P16473 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2200003 0.86 KMT2A (0.39) KMT2ABCHEKDM4EADRB2BLM
SCHEMBL2196598 0.80 ADRB2 (0.48) KMT2AKDM4EADRB2BLMLMNA
SCHEMBL5064328 0.78 KMT2A (0.41) KMT2AKDM4EADRB2BLMLMNA
SCHEMBL2198620 0.77 ADRB2 (0.44) KMT2ABCHEKDM4EADRB2BLM
SCHEMBL2200379 0.77 ADRB2 (0.44) KMT2ABCHEKDM4EADRB2BLM
SCHEMBL2197814 0.77 KDM4E (0.57) BCHEKDM4EADRB2LMNAADRB3
SCHEMBL2195384 0.76 RIPK1 (0.37) KMT2AKDM4ELMNAMEN1CYP3A4
SCHEMBL2196410 0.76 RIPK1 (0.37) KMT2AKDM4ELMNAMEN1CYP3A4
SCHEMBL2199004 0.74 BCHE (0.47) BCHEADRB2ADRB1ADRB3
SCHEMBL2197422 0.74 BCHE (0.47) BCHEADRB2ADRB1ADRB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7977336-B2 Aminopyrimidine derivatives as PLK1 inhibitors BANYU PHARMACEUTICAL CO. LTD (JP) 2011-07-12 US disclosed
EP-2116543-A1 NOVEL AMINOPYRIMIDINE DERIVATIVE AS PLK1 INHIBITOR BANYU PHARMACEUTICAL CO., LTD. (JP) 2009-11-11 EP disclosed