SCHEMBL21995872

SCHEMBL21995872

O=C(c1nn(-c2ccccc2)c2c1CC1(CC2)OCCO1)N1CCCCC1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 8/20 0.51
TMEM97 Q5BJF2 4/20 0.51
ALDH1A1 P00352 3/20 0.45
TSHR P16473 1/20 0.45
PIK3CD O00329 5/20 0.44
PIK3R2 O00459 5/20 0.44
PIK3CA P42336 5/20 0.44
PIK3CB P42338 5/20 0.44
PIK3CG P48736 5/20 0.44
PIK3R5 Q8WYR1 5/20 0.44
PIK3R3 Q92569 5/20 0.44
KDM4E B2RXH2 2/20 0.43
KMT2A Q03164 1/20 0.42
UGCG Q16739 3/20 0.41
USP2 O75604 1/20 0.41
LMNA P02545 1/20 0.41
POLB P06746 1/20 0.41
HPGD P15428 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21995870 0.82 SIGMAR1 (0.52) SIGMAR1TMEM97ALDH1A1TSHRPIK3CD
SCHEMBL27381184 0.78 SIGMAR1 (0.58) SIGMAR1TMEM97ALDH1A1TSHRPIK3CD
SCHEMBL8085636 0.77 GRIA2 (0.68)
SCHEMBL18209687 0.77 TMEM97 (0.49) SIGMAR1TMEM97ALDH1A1PIK3CDPIK3R2
SCHEMBL21995880 0.71 KMT2A (0.39) ALDH1A1TSHRKMT2ALMNAPOLB
SCHEMBL22049303 0.68 SIGMAR1 (0.73) SIGMAR1TMEM97PIK3CDPIK3R2PIK3CA
SCHEMBL22048884 0.67 SIGMAR1 (1.00) SIGMAR1TMEM97PIK3CDPIK3R2PIK3CA
SCHEMBL22049298 0.67 SIGMAR1 (1.00) SIGMAR1TMEM97ALDH1A1TSHRPIK3CD
SCHEMBL30936641 0.65 CNR1 (0.69) ALDH1A1TSHRPIK3CDPIK3R2PIK3CA
SCHEMBL24999576 0.65 SIGMAR1 (0.67) SIGMAR1TMEM97ALDH1A1KDM4EKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020112846-A1 SMALL MOLECULE MODULATORS OF SIGMA-1 AND SIGMA-2 RECEPTORS AND USES THEREOF NORTHWESTERN UNIVERSITY (US) 2020-06-04 WO disclosed