SCHEMBL21995870

SCHEMBL21995870

O=C(c1c2c(nn1-c1ccccc1)CCC1(C2)OCCO1)N1CCCCC1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 9/20 0.52
TMEM97 Q5BJF2 6/20 0.52
PIK3CD O00329 3/20 0.42
PIK3R2 O00459 3/20 0.42
PIK3CA P42336 3/20 0.42
PIK3CB P42338 3/20 0.42
PIK3CG P48736 3/20 0.42
PIK3R5 Q8WYR1 3/20 0.42
PIK3R3 Q92569 3/20 0.42
ALDH1A1 P00352 6/20 0.42
TSHR P16473 2/20 0.42
HPGD P15428 2/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
KDM4E B2RXH2 1/20 0.38
LMNA P02545 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
USP2 O75604 1/20 0.38
POLB P06746 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
CREBBP Q92793 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21995872 0.82 SIGMAR1 (0.51) SIGMAR1TMEM97PIK3CDPIK3R2PIK3CA
SCHEMBL8085636 0.68 GRIA2 (0.68)
SCHEMBL22048590 0.67 SIGMAR1 (0.72) SIGMAR1TMEM97PIK3CDPIK3R2PIK3CA
SCHEMBL22048598 0.67 SIGMAR1 (0.90) SIGMAR1TMEM97
SCHEMBL21995880 0.65 KMT2A (0.39) ALDH1A1TSHRHPGDLMNAPOLB
SCHEMBL29019285 0.65 ALDH1A1 (0.35) PIK3CDPIK3R2PIK3CAPIK3CBPIK3CG
SCHEMBL22048589 0.64 SIGMAR1 (0.84) SIGMAR1TMEM97
SCHEMBL18209687 0.63 TMEM97 (0.49) SIGMAR1TMEM97PIK3CDPIK3R2PIK3CA
SCHEMBL27381184 0.62 SIGMAR1 (0.58) SIGMAR1TMEM97PIK3CDPIK3R2PIK3CA
SCHEMBL24029478 0.62 OPRM1 (0.37) PIK3CDPIK3R2PIK3CAPIK3CBPIK3CG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020112846-A1 SMALL MOLECULE MODULATORS OF SIGMA-1 AND SIGMA-2 RECEPTORS AND USES THEREOF NORTHWESTERN UNIVERSITY (US) 2020-06-04 WO disclosed