SCHEMBL2200148

SCHEMBL2200148

Cc1ccc(-c2cc(F)ccc2NC(=O)c2sc(C)nc2C(F)(F)F)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 6/20 0.49
NPSR1 Q6W5P4 1/20 0.44
WDR5 P61964 1/20 0.44
GAA P10253 2/20 0.44
THRB P10828 1/20 0.41
KDM4E B2RXH2 2/20 0.40
HTT P42858 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
ALDH1A1 P00352 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2C19 P33261 1/20 0.40
F10 P00742 1/20 0.39
LMNA P02545 2/20 0.39
TP53 P04637 1/20 0.39
NTRK1 P04629 1/20 0.39
NTRK2 Q16620 1/20 0.39
RAB9A P51151 1/20 0.38
KMT2A Q03164 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4162627 0.89 MAPT (0.49) MAPTWDR5GAAKDM4EHTT
SCHEMBL2202643 0.88 CHRM3 (0.44) MAPTWDR5GAATHRBKDM4E
SCHEMBL2199612 0.87 CHRM3 (0.44) MAPTNPSR1WDR5GAATHRB
SCHEMBL12424051 0.87 WDR5 (0.41) MAPTWDR5GAATHRBKDM4E
SCHEMBL13210783 0.85 NTRK1 (0.51) MAPTWDR5GAATHRBKDM4E
SCHEMBL2199397 0.82 MEN1 (0.48) MAPTNPSR1WDR5GAATHRB
SCHEMBL13873513 0.82 MAPT (0.49) MAPTWDR5GAATHRBKDM4E
SCHEMBL2196885 0.81 LIPE (0.46) MAPTNPSR1WDR5GAATHRB
SCHEMBL4158657 0.81 MAPT (0.48) MAPTNPSR1WDR5GAATHRB
SCHEMBL14564515 0.80 MAPT (0.46) MAPTNPSR1WDR5GAAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7977363-B2 Fungicides/bactericides for plant protection; exhibit a strong fortifying effect in plants; for controlling cereal diseases against Puccinia species, and diseases in viticulture and fruit and vegetable production against Botrytis, Venturia or Alternaria species; low toxicity; tolrerance BAYER CROPSCIENCE AG (DE) 2011-07-12 US disclosed
US-20090105316-A1 Biphenyl Thiazole Carboxamides BAYER CROPSCIENCE AG (DE) 2009-04-23 US disclosed
US-20080242708-A1 Biphenyl-Thiazolo-Carboxamides BAYER CROPSCIENCE AG (DE) 2008-10-02 US disclosed
EP-1786794-A2 BIPHENYL-THIAZOLO-CARBOXAMIDES Bayer CropScience Aktiengesellschaft (DE) 2007-05-23 EP disclosed
WO-2006024387-A2 BIPHENYL-THIAZOLO-CARBOXAMIDES BAYER CROPSCIENCE AG (DE) 2006-03-09 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080242708-A1 Biphenyl-Thiazolo-Carboxamides MRPL21, CBR3, NAT1 MAPT 2387/4885NPSR1 1178/4885WDR5 1530/4885
US-20090105316-A1 Biphenyl Thiazole Carboxamides MRPL21, CBR3, BRD4 MAPT 2171/4885NPSR1 1857/4885WDR5 1277/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.