SCHEMBL22004377

SCHEMBL22004377

Cn1c(-c2ccc(OC(F)(F)F)cc2)cc2cc(Cl)ccc21

nearest known ligand 0.54

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ACLY P53396 6/20 0.54
F2RL3 Q96RI0 1/20 0.43
DHODH Q02127 1/20 0.41
HSD11B1 P28845 1/20 0.41
MARS1 P56192 1/20 0.40
CYP3A4 P08684 1/20 0.40
CCR6 P51684 3/20 0.39
KMT2A Q03164 2/20 0.39
MEN1 O00255 1/20 0.39
LMNA P02545 1/20 0.39
MAPK1 P28482 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
CHRNA7 P36544 1/20 0.38
GRIN2B Q13224 1/20 0.38
KCNH2 Q12809 1/20 0.38
ALOX5 P09917 1/20 0.38
PTGES O14684 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22004110 0.86 ACLY (0.57) ACLYF2RL3HSD11B1KMT2APTGES
SCHEMBL22004376 0.83 ACLY (0.52) ACLYDHODHHSD11B1MARS1CYP3A4
SCHEMBL22021620 0.83 ACLY (0.50) ACLYCYP3A4KMT2ASMN1; SMN2
SCHEMBL7799883 0.82 KMT2A (0.50) ACLYHSD11B1KMT2AMEN1LMNA
SCHEMBL22004165 0.81 ACLY (0.55) ACLYF2RL3CYP3A4PTGES
SCHEMBL22022198 0.81 ACLY (0.55) ACLYF2RL3
SCHEMBL8942357 0.76 KMT2A (0.66) ACLYKMT2AMEN1
SCHEMBL22004314 0.75 ACLY (0.51) ACLYF2RL3KMT2AKCNH2
SCHEMBL22004394 0.74 KCNH2 (0.48) ACLYKMT2AMEN1KCNH2
SCHEMBL22004328 0.73 ACLY (0.53) ACLYKMT2AMAPK1PTGES

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20200157076-A1 ACLY INHIBITORS AND USES THEREOF NIMBUS DISCOVERY, INC. 2020-05-21 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200157076-A1 ACLY INHIBITORS AND USES THEREOF ACLY, ATP5ME, ATP5MG ACLY 1/4885F2RL3 4563/4885DHODH 219/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.