SCHEMBL22005102

SCHEMBL22005102

Cc1c(-c2ccccc2)n(C(C)C)c2ccc(Cl)cc12

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACLY P53396 1/20 0.46
PTGS2 P35354 3/20 0.43
GRIK2 Q13002 1/20 0.40
TACR1 P25103 1/20 0.40
KDM4E B2RXH2 3/20 0.40
MAPT P10636 2/20 0.39
THRB P10828 1/20 0.39
PTGDR2 Q9Y5Y4 2/20 0.39
HCRTR1 O43613 1/20 0.38
CASP1 P29466 1/20 0.38
CASP7 P55210 1/20 0.38
EGFR P00533 2/20 0.37
PGR P06401 1/20 0.36
NR1I2 O75469 1/20 0.36
ADRA2A P08913 1/20 0.36
ADORA3 P0DMS8 1/20 0.36
TBXA2R P21731 1/20 0.36
OPRD1 P41143 1/20 0.36
PDE4D Q08499 1/20 0.36
PLA2G4A P47712 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22003801 0.81 PTGDR2 (0.45) ACLYKDM4EMAPTTHRBPTGDR2
SCHEMBL22005104 0.80 KDM4E (0.50) ACLYPTGS2GRIK2TACR1KDM4E
SCHEMBL22004308 0.78 RAB9A (0.48) ACLYKDM4EMAPTTHRBPTGDR2
SCHEMBL13222023 0.75 MAPT (0.51) PTGS2MAPTTHRBPTGDR2HTT
SCHEMBL11601877 0.72 CASR (0.67) PTGS2EGFRNR1I2ADRA2AADORA3
SCHEMBL22004380 0.72 ACLY (0.58) ACLYKDM4EMAPTPTGDR2PLA2G4A
SCHEMBL9539031 0.70 KDM4E (0.44) KDM4EMAPTCASP1CASP7RAB9A
SCHEMBL9539113 0.70 KDM4E (0.48) PTGS2KDM4EMAPTCASP1CASP7
SCHEMBL22003798 0.70 ACLY (0.44) ACLYMAPTTHRB
SCHEMBL29839883 0.70 ACLY (0.64) ACLYPTGS2LMNAL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020102616-A1 ACLY INHIBITORS AND USES THEREOF Nimbus Artemis, Inc. (US) 2020-05-22 WO disclosed
US-20200157076-A1 ACLY INHIBITORS AND USES THEREOF NIMBUS DISCOVERY, INC. 2020-05-21 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200157076-A1 ACLY INHIBITORS AND USES THEREOF ACLY, ATP5ME, ATP5MG ACLY 1/4885PTGS2 4122/4885GRIK2 1910/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.