SCHEMBL220117

SCHEMBL220117

Cc1ccn[nH]1.Clc1cc(Cl)nc(Cl)n1

nearest known ligand 0.37

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HPGDS O60760 2/20 0.37
PLK4 O00444 1/20 0.35
PAK4 O96013 1/20 0.35
NOTUM Q6P988 2/20 0.34
COMT P21964 2/20 0.33
POLB P06746 1/20 0.33
PTPN11 Q06124 1/20 0.33
ALDH1A1 P00352 2/20 0.33
PIM1 P11309 1/20 0.33
PDPK1 O15530 1/20 0.31
PIK3C3 Q8NEB9 1/20 0.31
LMNA P02545 2/20 0.31
KDM4E B2RXH2 2/20 0.31
RECQL P46063 1/20 0.31
KMT2A Q03164 1/20 0.31
MAPK1 P28482 1/20 0.30
NPC1 O15118 1/20 0.30
RAB9A P51151 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL45219 0.78
SCHEMBL218052 0.71
Ammonia Solution, Strong SCHEMBL27915759 0.71 ALDH1A1 (0.50) ALDH1A1LMNAKDM4EKMT2A
SCHEMBL8621552 0.69 HPGDS (0.36) HPGDSCOMTPOLBPTPN11ALDH1A1
Methyl Alcohol SCHEMBL29141832 0.69 ALDH1A1 (0.41) POLBALDH1A1LMNAKDM4EKMT2A
SCHEMBL9978274 0.65 TSHR (0.43) NOTUMPOLBKDM4EKMT2ANPC1
SCHEMBL30350717 0.65
SCHEMBL104786 0.65
Formaldehyde SCHEMBL27883709 0.64 ALDH1A1 (0.41) ALDH1A1LMNAKMT2A
SCHEMBL341468 0.63 PIK3C3 (0.44) ALDH1A1PIK3C3KDM4EKMT2AMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8088784-B2 4-(3-aminopyrazole) pyrimidine derivatives for use as tyrosine kinase inhibitors in the treatment of cancer ASTRAZENECA AB (SE) 2012-01-03 US disclosed