SCHEMBL22011829

SCHEMBL22011829

CC(=O)N=S(N)(=O)c1ccc(C(C)(C)O)cc1F

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 1/20 0.35
NR1H4 Q96RI1 1/20 0.35
CA2 P00918 8/20 0.35
CA1 P00915 5/20 0.35
CA9 Q16790 3/20 0.35
AKR1C3 P42330 1/20 0.34
AKR1C2 P52895 1/20 0.34
HSD11B1 P28845 6/20 0.33
ABCC9 O60706 1/20 0.33
ABCC8 Q09428 1/20 0.33
KCNJ11 Q14654 1/20 0.33
KCNJ8 Q15842 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
NR1I2 O75469 1/20 0.33
CA4 P22748 1/20 0.32
CA12 O43570 1/20 0.32
PTGS1 P23219 1/20 0.32
PTGS2 P35354 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22013719 0.89 AKR1C3 (0.34) EPHX2NR1H4CA2CA1AKR1C3
SCHEMBL20698926 0.84 CA2 (0.34) EPHX2NR1H4CA2CA1CA9
SCHEMBL29927632 0.80 CA2 (0.41) EPHX2NR1H4CA2CA1HSD11B1
SCHEMBL19507908 0.80 CA2 (0.41) EPHX2NR1H4CA2CA1HSD11B1
SCHEMBL20680978 0.79 APLNR (0.33) EPHX2NR1H4CA2AKR1C3AKR1C2
SCHEMBL25033452 0.76 NLRP3 (0.38) CA2
SCHEMBL30243978 0.76 NLRP3 (0.38) CA2
SCHEMBL21892944 0.76 NLRP3 (0.38) CA2
SCHEMBL20692357 0.76 NLRP3 (0.38) CA2
SCHEMBL21810663 0.76 NLRP3 (0.47) CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020102576-A1 COMPOUNDS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH NLRP ACTIVITY NOVARTIS INFLAMMASOME RESEARCH, INC. (US) 2020-05-22 WO disclosed