SCHEMBL22012064

SCHEMBL22012064

CN(Cc1ccc([S+](N)[O-])c(F)c1)C(=O)OC(C)(C)C

nearest known ligand 0.36

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 5/20 0.36
SLC6A4 P31645 5/20 0.36
GRM2 Q14416 1/20 0.36
GLS O94925 2/20 0.36
RIPK1 Q13546 3/20 0.36
CACNA1G O43497 1/20 0.35
CACNA1B Q00975 1/20 0.35
CACNA1C Q13936 1/20 0.35
HTR2A P28223 1/20 0.35
P2RY1 P47900 1/20 0.33
MGLL Q99685 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18416938 0.79 SSTR4 (0.40) HTR2CSLC6A4GRM2GLSRIPK1
SCHEMBL20692404 0.78 HTR2C (0.38) HTR2CSLC6A4GRM2GLSRIPK1
SCHEMBL30244191 0.78 HTR2C (0.38) HTR2CSLC6A4GRM2GLSRIPK1
SCHEMBL506105 0.78 RIPK1 (0.40) HTR2CSLC6A4GRM2GLSRIPK1
SCHEMBL506457 0.77 GRM2 (0.40) HTR2CSLC6A4GRM2GLSRIPK1
SCHEMBL20692405 0.76 HTR2C (0.39) HTR2CSLC6A4GRM2GLSRIPK1
SCHEMBL22012402 0.76 HRH3 (0.38) P2RY1
SCHEMBL7430459 0.75 RIPK1 (0.59) HTR2CSLC6A4GRM2RIPK1HTR2A
SCHEMBL506166 0.74 HTR2C (0.36) HTR2CSLC6A4GRM2GLSRIPK1
SCHEMBL506165 0.74 HTR2C (0.36) HTR2CSLC6A4GRM2GLSRIPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020102576-A1 COMPOUNDS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH NLRP ACTIVITY NOVARTIS INFLAMMASOME RESEARCH, INC. (US) 2020-05-22 WO disclosed