SCHEMBL22012074

SCHEMBL22012074

CC(C)(C)[Si](C)(C)N=S(N)(=O)c1cc2c(s1)CCNC2

nearest known ligand 0.43

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PNMT P11086 9/20 0.43
ADRA2A P08913 1/20 0.36
ADRA2B P18089 1/20 0.36
ADRA2C P18825 1/20 0.36
PARP1 P09874 3/20 0.32
PARP2 Q9UGN5 3/20 0.32
KCNH2 Q12809 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22012907 0.82 FBP1 (0.41)
SCHEMBL22012118 0.79 PARP1 (0.36) PARP1PARP2
SCHEMBL6673498 0.76 PNMT (0.54) PNMTADRA2AADRA2BADRA2CPARP1
Hydrochloric Acid SCHEMBL21962263 0.75 PNMT (0.53) PNMTADRA2AADRA2BADRA2CPARP1
SCHEMBL30244132 0.74 PNMT (0.51) PNMTADRA2AADRA2BADRA2CPARP1
SCHEMBL21962438 0.73 PRMT5 (0.32)
SCHEMBL22012113 0.72 NR1H2 (0.45)
SCHEMBL25031530 0.69 KDM4D (0.32)
SCHEMBL23569183 0.69 PTGES2 (0.40)
SCHEMBL20692370 0.67

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020102576-A1 COMPOUNDS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH NLRP ACTIVITY NOVARTIS INFLAMMASOME RESEARCH, INC. (US) 2020-05-22 WO disclosed