SCHEMBL22012199

SCHEMBL22012199

C=NCc1cc(C(C)C)c(NC(=O)N=S(N)(=O)c2ccc(S(C)(=O)=O)cc2)c(C(C)C)c1

nearest known ligand 0.33

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NLRP3 Q96P20 3/20 0.33
HSP90AA1 P07900 5/20 0.32
CA12 O43570 2/20 0.32
CA1 P00915 2/20 0.32
CA2 P00918 2/20 0.32
CA9 Q16790 2/20 0.32
HSP90B1 P14625 1/20 0.32
TRAP1 Q12931 1/20 0.32
TGM2 P21980 1/20 0.32
HSP90AB1 P08238 1/20 0.32
RORC P51449 1/20 0.31
SLC9A1 P19634 1/20 0.31
GRIN2B Q13224 1/20 0.31
POLB P06746 1/20 0.31
PSMB5 P28074 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25033764 0.84 NLRP3 (0.40) NLRP3HSP90AA1CA12CA1CA2
SCHEMBL20692355 0.83 NLRP3 (0.35) NLRP3HSP90AA1CA12CA1CA2
SCHEMBL26009908 0.83 NLRP3 (0.35) NLRP3HSP90AA1CA12CA1CA2
SCHEMBL23481741 0.83 NLRP3 (0.35) NLRP3HSP90AA1CA12CA1CA2
SCHEMBL20692181 0.82 CA2 (0.36) NLRP3HSP90AA1CA12CA1CA2
SCHEMBL20692406 0.81 PTGDR2 (0.38) NLRP3HSP90AA1CA12CA1CA2
SCHEMBL30244043 0.81 PTGDR2 (0.38) NLRP3HSP90AA1CA12CA1CA2
SCHEMBL30243773 0.81 PTGDR2 (0.38) NLRP3HSP90AA1CA12CA1CA2
SCHEMBL22013424 0.76 NLRP3 (0.35) NLRP3
SCHEMBL22012200 0.75 CA2 (0.37) NLRP3CA12CA1CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020102576-A1 COMPOUNDS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH NLRP ACTIVITY NOVARTIS INFLAMMASOME RESEARCH, INC. (US) 2020-05-22 WO disclosed