SCHEMBL22012833

SCHEMBL22012833

Oc1ccc(CC2N=N2)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 4/20 0.48
ESR2 Q92731 2/20 0.48
ABAT P80404 1/20 0.44
CAPN1 P07384 1/20 0.44
CA2 P00918 3/20 0.42
TAAR1 Q96RJ0 4/20 0.41
SLC6A2 P23975 2/20 0.41
KDM4E B2RXH2 2/20 0.41
ALDH1A1 P00352 2/20 0.41
IDO1 P14902 2/20 0.41
HTR1A P08908 1/20 0.41
ADRA2A P08913 1/20 0.41
CYP2C19 P33261 1/20 0.41
HTR3A P46098 1/20 0.41
BACE1 P56817 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
BLM P54132 2/20 0.40
KMT2A Q03164 2/20 0.40
MEN1 O00255 1/20 0.40
NPC1 O15118 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22013139 0.77 CYP3A4 (0.41) IDO1CYP3A4PMP22
SCHEMBL18909585 0.75 TP53 (0.42) CA2TAAR1ALDH1A1CYP2C19L3MBTL1
SCHEMBL16902819 0.70 GRIN2B (0.49) ESR1ESR2CYP3A4
SCHEMBL14734507 0.70 GRIN2B (0.49) ESR1ESR2CYP3A4
SCHEMBL12290753 0.67 ESR1 (0.50) ESR1ESR2ALDH1A1KMT2ANPC1
SCHEMBL21155257 0.67 ESR1 (0.44) ESR1ESR2ABATCAPN1CA2
SCHEMBL5522519 0.67 ALOX5 (0.45) ESR1ESR2ABATCAPN1CA2
SCHEMBL10824285 0.67 CAPN1 (0.46) ESR1ESR2ABATCAPN1CA2
SCHEMBL13472627 0.67 ESR1 (0.44) ESR1ESR2ABATCAPN1CA2
SCHEMBL2969737 0.66 ESR1 (1.00) ESR1ESR2ABATCA2TAAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20220098155-A1 NOVEL PATHWAY FOR THE SYNTHESIS OF DIAZIRINES, THAT MAY OR MAY NOT BE ENRICHED IN NITROGEN-15 INSTITUT NATIONAL DES SCIENCES APPLIQUEES DE ROUEN (INSA) (FR) 2022-03-31 US disclosed
WO-2020099596-A1 NOVEL PATHWAY FOR THE SYNTHESIS OF DIAZIRINES, THAT MAY OR MAY NOT BE ENRICHED IN NITROGEN-15 UNIVERSITE DE ROUEN NORMANDIE (FR) 2020-05-22 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220098155-A1 NOVEL PATHWAY FOR THE SYNTHESIS OF DIAZIRINES, THAT MAY OR MAY NOT BE ENRICHED IN NITROGEN-15 SSTR5, SLC6A15, SLC1A5 ESR1 3129/4885ESR2 3521/4885ABAT 617/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.