SCHEMBL22012952

SCHEMBL22012952

C=CCc1c2c(c(NC(N)=O)c3c1CCC3)CCC2

nearest known ligand 0.33

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.33
CYP1A2 P05177 1/20 0.31
KDM4E B2RXH2 1/20 0.30
MAPK1 P28482 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22012961 0.75 KDM4E (0.40) GAACYP1A2KDM4EMAPK1
SCHEMBL21962269 0.72 ACHE (0.35) MAPK1
SCHEMBL21646660 0.71 ALDH1A1 (0.36) GAACYP1A2KDM4EMAPK1
SCHEMBL25842067 0.71 NLRP3 (0.37) GAACYP1A2KDM4EMAPK1
SCHEMBL22012481 0.67 POLB (0.40) GAAKDM4E
SCHEMBL18029669 0.66 NLRP3 (0.53)
SCHEMBL22019806 0.66 GAA (0.59) GAACYP1A2KDM4EMAPK1
SCHEMBL29494713 0.65 NLRP3 (0.51)
Potassium SCHEMBL29676171 0.65 NLRP3 (0.51)
SCHEMBL25845405 0.65 NLRP3 (0.51)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020102576-A1 COMPOUNDS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH NLRP ACTIVITY NOVARTIS INFLAMMASOME RESEARCH, INC. (US) 2020-05-22 WO disclosed