SCHEMBL22013114

SCHEMBL22013114

CSn1cc(-c2c(Cl)cnc3ccc(N4CCC(F)C4)nc23)cn1

nearest known ligand 0.37

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
MAP4K4 O95819 8/20 0.37
LRRK2 Q5S007 5/20 0.37
P2RX7 Q99572 4/20 0.34
MELK Q14680 3/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23836958 1.00 MAP4K4 (0.37) MAP4K4LRRK2P2RX7MELK
SCHEMBL23836972 0.90 MAP4K4 (0.37) MAP4K4LRRK2P2RX7MELK
SCHEMBL23837007 0.88 LRRK2 (0.45) MAP4K4LRRK2
SCHEMBL22014126 0.83 KHK (0.39) MAP4K4LRRK2P2RX7MELK
SCHEMBL23837054 0.83 MAP4K4 (0.36) MAP4K4LRRK2P2RX7MELK
SCHEMBL23836989 0.82 MELK (0.41) MAP4K4LRRK2MELK
SCHEMBL22013423 0.81 KHK (0.37) MAP4K4LRRK2P2RX7
SCHEMBL23837072 0.81 FGFR1 (0.37) MAP4K4LRRK2P2RX7MELK
SCHEMBL23836970 0.81 FGFR1 (0.37) MAP4K4LRRK2P2RX7MELK
SCHEMBL23837050 0.81 P2RX7 (0.39) MAP4K4LRRK2P2RX7MELK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020098723-A1 SIX-MEMBERED AND SIX-MEMBERED HETEROCYCLIC COMPOUND AND USES THEREOF SERVING AS PROTEIN RECEPTOR KINASE INHIBITOR 上海轶诺药业有限公司 2020-05-22 WO disclosed