SCHEMBL22013423

SCHEMBL22013423

FC1CCN(c2ccc3ncc(Cl)c(-c4cnn(C5CNC5)c4)c3n2)C1

nearest known ligand 0.37

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
KHK P50053 3/20 0.37
MET P08581 3/20 0.37
MAP4K4 O95819 3/20 0.36
P2RX7 Q99572 6/20 0.35
LRRK2 Q5S007 1/20 0.33
PTPN11 Q06124 4/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23836949 0.94 MET (0.40) KHKMETLRRK2
SCHEMBL23836963 0.92 MET (0.41) KHKMETMAP4K4P2RX7
SCHEMBL22013656 0.92 CHRNA4 (0.40) KHKMETLRRK2
SCHEMBL23837041 0.90 MAP4K4 (0.36) KHKMETMAP4K4LRRK2
SCHEMBL23836974 0.90 MAP4K4 (0.36) KHKMETMAP4K4LRRK2
SCHEMBL22014126 0.89 KHK (0.39) KHKMAP4K4P2RX7LRRK2
SCHEMBL23836989 0.88 MELK (0.41) METMAP4K4LRRK2
SCHEMBL23837009 0.86 P2RX7 (0.39) MAP4K4P2RX7LRRK2
SCHEMBL23837050 0.86 P2RX7 (0.39) MAP4K4P2RX7LRRK2
SCHEMBL23837042 0.86 MAP4K4 (0.34) MAP4K4P2RX7LRRK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3882247-A1 SIX-MEMBERED AND SIX-MEMBERED HETEROCYCLIC COMPOUND AND USES THEREOF SERVING AS PROTEIN RECEPTOR KINASE INHIBITOR Shanghai Ennovabio Pharmaceuticals Co., Ltd. (CN) 2021-09-22 EP disclosed
WO-2020098723-A1 SIX-MEMBERED AND SIX-MEMBERED HETEROCYCLIC COMPOUND AND USES THEREOF SERVING AS PROTEIN RECEPTOR KINASE INHIBITOR 上海轶诺药业有限公司 2020-05-22 WO disclosed