SCHEMBL22014126

SCHEMBL22014126

CN1CC(n2cc(-c3c(Cl)cnc4ccc(N5CCC(F)C5)nc34)cn2)C1

nearest known ligand 0.39

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
KHK P50053 3/20 0.39
LRRK2 Q5S007 3/20 0.36
MAP4K4 O95819 7/20 0.36
MELK Q14680 4/20 0.34
P2RX7 Q99572 3/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23836989 0.94 MELK (0.41) LRRK2MAP4K4MELK
SCHEMBL22013423 0.89 KHK (0.37) KHKLRRK2MAP4K4P2RX7
SCHEMBL23837007 0.88 LRRK2 (0.45) LRRK2MAP4K4
SCHEMBL23837009 0.88 P2RX7 (0.39) LRRK2MAP4K4MELKP2RX7
SCHEMBL23837050 0.88 P2RX7 (0.39) LRRK2MAP4K4MELKP2RX7
SCHEMBL22013656 0.88 CHRNA4 (0.40) KHKLRRK2
SCHEMBL23836949 0.86 MET (0.40) KHKLRRK2
SCHEMBL23837042 0.86 MAP4K4 (0.34) LRRK2MAP4K4MELKP2RX7
SCHEMBL23836952 0.86 MET (0.39) KHKMELKP2RX7
SCHEMBL22013265 0.86 P2RX7 (0.34) LRRK2MAP4K4P2RX7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3882247-A1 SIX-MEMBERED AND SIX-MEMBERED HETEROCYCLIC COMPOUND AND USES THEREOF SERVING AS PROTEIN RECEPTOR KINASE INHIBITOR Shanghai Ennovabio Pharmaceuticals Co., Ltd. (CN) 2021-09-22 EP disclosed
WO-2020098723-A1 SIX-MEMBERED AND SIX-MEMBERED HETEROCYCLIC COMPOUND AND USES THEREOF SERVING AS PROTEIN RECEPTOR KINASE INHIBITOR 上海轶诺药业有限公司 2020-05-22 WO disclosed