SCHEMBL22013956

SCHEMBL22013956

C[Si](C)(C)CCOCn1nc(Br)c2cc(Cl)cnc21

nearest known ligand 0.36

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 3/20 0.36
NPC1 O15118 1/20 0.30
MAPT P10636 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29511367 1.00 DGAT1 (0.36) DGAT1NPC1MAPT
SCHEMBL19023210 0.86 SPR (0.36) DGAT1NPC1MAPT
SCHEMBL19250755 0.85 NPC1 (0.32) DGAT1NPC1MAPT
SCHEMBL30908091 0.81 NPC1 (0.39) DGAT1NPC1MAPT
SCHEMBL30908064 0.80 MAPT (0.37) DGAT1NPC1MAPT
SCHEMBL1592603 0.80 MAPT (0.37) DGAT1NPC1MAPT
SCHEMBL22553893 0.80 DGAT1 (0.35) DGAT1MAPT
SCHEMBL22013944 0.79 NPC1 (0.37) DGAT1NPC1MAPT
SCHEMBL30908117 0.79 NPC1 (0.37) DGAT1NPC1MAPT
SCHEMBL30908118 0.79 NPC1 (0.37) DGAT1NPC1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3919490-A1 FIVE-AND-SIX-MEMBERED HETEROCYCLIC COMPOUND AND USE THEREOF AS PROTEIN RECEPTOR KINASE INHIBITOR Shanghai Ennovabio Pharmaceuticals Co., Ltd. (CN) 2021-12-08 EP disclosed
WO-2020098720-A1 FIVE-AND-SIX-MEMBERED HETEROCYCLIC COMPOUND AND USE THEREOF AS PROTEIN RECEPTOR KINASE INHIBITOR 上海轶诺药业有限公司 2020-05-22 WO disclosed