SCHEMBL29511367

SCHEMBL29511367

C[Si](C)(C)CCOCn1nc(Br)c2cc(Cl)cnc21

nearest known ligand 0.36

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 3/20 0.36
NPC1 O15118 1/20 0.30
MAPT P10636 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22013956 1.00 DGAT1 (0.36) DGAT1NPC1MAPT
SCHEMBL19023210 0.86 SPR (0.36) DGAT1NPC1MAPT
SCHEMBL19250755 0.85 NPC1 (0.32) DGAT1NPC1MAPT
SCHEMBL30908091 0.81 NPC1 (0.39) DGAT1NPC1MAPT
SCHEMBL30908064 0.80 MAPT (0.37) DGAT1NPC1MAPT
SCHEMBL1592603 0.80 MAPT (0.37) DGAT1NPC1MAPT
SCHEMBL22553893 0.80 DGAT1 (0.35) DGAT1MAPT
SCHEMBL22013944 0.79 NPC1 (0.37) DGAT1NPC1MAPT
SCHEMBL30908117 0.79 NPC1 (0.37) DGAT1NPC1MAPT
SCHEMBL30908118 0.79 NPC1 (0.37) DGAT1NPC1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12391687-B2 Five-and-six-membered heterocyclic compound and use thereof as protein receptor kinase inhibitor SHANGHAI ENNOVABIO PHARMACEUTICALS CO., LTD. (CN) 2025-08-19 US disclosed
EP-3919490-B1 FIVE-AND-SIX-MEMBERED HETEROCYCLIC COMPOUND AND USE THEREOF AS PROTEIN RECEPTOR KINASE INHIBITOR SHANGHAI ENNOVABIO PHARMACEUTICALS CO LTD (CN) 2025-04-02 EP disclosed
CN-113166142-B Five-membered and six-membered heterocyclic compounds and application thereof as protein receptor kinase inhibitors 上海轶诺药业有限公司 2024-04-26 CN disclosed
US-20220144827-A1 FIVE-AND-SIX-MEMBERED HETEROCYCLIC COMPOUND AND USE THEREOF AS PROTEIN RECEPTOR KINASE INHIBITOR SHANGHAI ENNOVABIO PHARMACEUTICALS CO., LTD. (CN) 2022-05-12 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12391687-B2 Five-and-six-membered heterocyclic compound and use thereof as protein receptor kinase inhibitor GRK6, GRK3, ERBB2 DGAT1 3470/4885NPC1 2977/4885MAPT 2101/4885
US-20220144827-A1 FIVE-AND-SIX-MEMBERED HETEROCYCLIC COMPOUND AND USE THEREOF AS PROTEIN RECEPTOR KINASE INHIBITOR GRK6, GRK3, ERBB2 DGAT1 3470/4885NPC1 2977/4885MAPT 2101/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.