SCHEMBL22014300

SCHEMBL22014300

COC(=O)C1(CC(C)C)CCN(C)CC1

nearest known ligand 0.37

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 1/20 0.36
CYP4F2 P78329 1/20 0.36
CYP4A11 Q02928 1/20 0.36
OPRM1 P35372 6/20 0.34
KCNH2 Q12809 2/20 0.34
SLC22A1 O15245 1/20 0.34
SLC6A4 P31645 1/20 0.34
ADRA1A P35348 1/20 0.34
OPRD1 P41143 1/20 0.34
OPRK1 P41145 1/20 0.34
CYP2C19 P33261 1/20 0.33
SCN1A P35498 1/20 0.33
SCN2A Q99250 1/20 0.33
SCN3A Q9NY46 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13199857 0.85 CYP4F2 (0.46) CYP2D6CYP4F2CYP4A11CYP2C19
SCHEMBL379072 0.83 OPRM1 (0.48) OPRM1KCNH2SLC22A1SLC6A4ADRA1A
SCHEMBL13715140 0.82 CYP4F2 (0.47) CYP2D6CYP4F2CYP4A11CYP2C19
SCHEMBL16508898 0.80 OPRM1 (0.40) CYP4F2CYP4A11OPRM1KCNH2SLC22A1
SCHEMBL19483314 0.79 CYP2C19 (0.32) CYP2C19
SCHEMBL89520 0.77 PKM (0.47) CYP2D6CYP4F2CYP4A11
SCHEMBL22014531 0.77 CYP4F2 (0.44) CYP4F2CYP4A11OPRM1KCNH2SLC22A1
SCHEMBL12540731 0.76 MAPK1 (0.46) CYP4F2CYP4A11OPRM1KCNH2SLC22A1
SCHEMBL22014295 0.73 SCN1A (0.36) CYP2D6OPRM1KCNH2SLC22A1SLC6A4
SCHEMBL20446734 0.72 MEN1 (0.34) CYP2D6CYP4F2CYP4A11CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020099885-A1 HETEROCYCLIC SPIRO-COMPOUNDS AS AM2 RECEPTOR INHIBITORS THE UNIVERSITY OF SHEFFIELD (GB) 2020-05-22 WO disclosed