SCHEMBL22014365

SCHEMBL22014365

CC(C)c1cc2c(c(C(C)C)c1CC(=O)NN)OC(F)(F)O2

nearest known ligand 0.38

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NLRP3 Q96P20 2/20 0.38
SOAT2 O75908 1/20 0.32
MYC P01106 1/20 0.32
SOAT1 P35610 1/20 0.32
MAP2K3 P46734 1/20 0.32
GABRA1 P14867 1/20 0.31
GABRG2 P18507 1/20 0.31
GABRB3 P28472 1/20 0.31
ADORA3 P0DMS8 1/20 0.30
ADORA2A P29274 1/20 0.30
ADORA2B P29275 1/20 0.30
ADORA1 P30542 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22014739 0.86 NLRP3 (0.33) NLRP3GABRA1GABRG2GABRB3
SCHEMBL30276820 0.86 NLRP3 (0.33) NLRP3GABRA1GABRG2GABRB3
SCHEMBL21962160 0.85 KDM4E (0.33) NLRP3GABRA1GABRG2GABRB3
SCHEMBL21962238 0.84 NLRP3 (0.33) NLRP3GABRA1GABRG2GABRB3
SCHEMBL25067068 0.70 NLRP3 (0.39) NLRP3
SCHEMBL25067070 0.70 NLRP3 (0.39) NLRP3
SCHEMBL16843335 0.67
SCHEMBL20028908 0.67 GABRA1 (0.30) GABRA1GABRG2GABRB3
SCHEMBL8859174 0.66 FABP3 (0.33)
SCHEMBL24192685 0.65 ADORA2A (0.34) ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020102574-A1 THE COMPOUNDS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH NLRP ACTIVITY NOVARTIS INFLAMMASOME RESEARCH, INC. (US) 2020-05-22 WO disclosed